SCHEMBL6640382

SCHEMBL6640382

CCCOc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1-c1nc2c(CCC)c(Cl)n(C)c2c(=O)[nH]1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 20/20 0.73
PDE6C P51160 3/20 0.68
PDE11A Q9HCR9 2/20 0.68
PDE6D O43924 2/20 0.65
PDE6A P16499 2/20 0.65
PDE6G P18545 2/20 0.65
PDE6B P35913 2/20 0.65
PDE6H Q13956 2/20 0.65
PDE2A O00408 1/20 0.65
ABCC4 O15439 1/20 0.65
ABCC5 O15440 1/20 0.65
PDE8A O60658 1/20 0.65
PDE9A O76083 1/20 0.65
ABCB11 O95342 1/20 0.65
CYP3A4 P08684 1/20 0.65
HTR1A P08908 1/20 0.65
PDE4A P27815 1/20 0.65
ADORA2A P29274 1/20 0.65
ADORA1 P30542 1/20 0.65
ADRA1A P35348 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6643884 0.94 PDE5A (0.73) PDE5APDE6CPDE11APDE6DPDE6A
SCHEMBL6647593 0.92 PDE5A (0.74) PDE5APDE1APDE1BPDE3BPDE1C
SCHEMBL6646009 0.92 PDE5A (0.65) PDE5APDE3BPDE3A
SCHEMBL6647256 0.91 PDE5A (0.73) PDE5APDE6CPDE11APDE6DPDE6A
SCHEMBL6643648 0.90 PDE5A (0.68) PDE5APDE3BPDE3A
SCHEMBL6646139 0.88 PDE5A (0.54) PDE5A
SCHEMBL6641363 0.87 PDE5A (0.74) PDE5APDE6CPDE11APDE6DPDE6A
SCHEMBL6646085 0.86 PDE5A (0.75) PDE5APDE6CPDE11APDE6DPDE6A
SCHEMBL6643499 0.86 PDE5A (0.65) PDE5APDE6CPDE11APDE6DPDE6A
SCHEMBL6643219 0.85 PDE5A (0.63) PDE5APDE6CPDE11APDE6DPDE6A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1257553-B1 PYRROLOPYRIMIDINONE DERIVATIVES, PROCESS OF PREPARATION AND USE SK CHEMICALS CO LTD (KR) 2004-05-26 EP disclosed