SCHEMBL6640464

SCHEMBL6640464

COc1cc(-c2cc(-c3ccnc(N)n3)ccc2O)nc(N)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.48
ALDH1A1 P00352 1/20 0.48
RAB9A P51151 1/20 0.48
AURKA O14965 2/20 0.45
PDPK1 O15530 2/20 0.45
TGFBR1 P36897 2/20 0.45
ROCK1 Q13464 2/20 0.45
AURKB Q96GD4 2/20 0.45
KMO O15229 1/20 0.45
CDK2 P24941 8/20 0.45
CDK1 P06493 6/20 0.45
CDK5 Q00535 2/20 0.43
CDK5R1 Q15078 2/20 0.43
CCNT1 O60563 3/20 0.42
CDK9 P50750 3/20 0.42
DYRK1A Q13627 2/20 0.42
DYRK3 O43781 1/20 0.42
DYRK2 Q92630 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
CCNA2 P20248 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6638867 0.84 CDK1 (0.58) NPC1ALDH1A1RAB9AAURKAPDPK1
SCHEMBL6640518 0.83 CDK1 (0.51) ALDH1A1AURKAPDPK1TGFBR1ROCK1
SCHEMBL6637999 0.83 NPC1 (0.51) NPC1ALDH1A1RAB9AAURKAPDPK1
SCHEMBL6638558 0.83 KMO (0.50) NPC1ALDH1A1RAB9AAURKAPDPK1
SCHEMBL6643177 0.81 KMO (0.55) AURKAPDPK1TGFBR1ROCK1AURKB
SCHEMBL7118870 0.79 CDK1 (0.48) NPC1ALDH1A1RAB9AAURKAPDPK1
SCHEMBL7112005 0.77 CCNT1 (0.42) NPC1ALDH1A1RAB9AAURKAPDPK1
SCHEMBL6642591 0.75 CDK1 (0.50) NPC1ALDH1A1RAB9AAURKAPDPK1
SCHEMBL6641629 0.75 CDK1 (0.50) NPC1ALDH1A1RAB9AAURKAPDPK1
SCHEMBL6638621 0.74 CDK1 (0.53) NPC1AURKAPDPK1KMOCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1412327-A2 INHIBITORS OF PROTEIN KINASE FOR THE TREATMENT OF DISEASE LG Biomedical Institute (US) 2004-04-28 EP claimed
US-20030187007-A1 Inhibitors of protein kinase for the treatment of disease LG BIOMEDICAL INSTITUTE 2003-10-02 US claimed
WO-2002096867-A2 INHIBITORS OF PROTEIN KINASE FOR THE TREATMENT OF DISEASE LG BIOMEDICAL INSTITUTE (US) 2002-12-05 WO claimed
US-20030208067-A1 Inhibitors of protein kinase for the treatment of disease LG BIOMEDICAL INSTITUTE 2003-11-06 US disclosed
US-20030187007-A1 Inhibitors of protein kinase for the treatment of disease LG BIOMEDICAL INSTITUTE 2003-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030208067-A1 Inhibitors of protein kinase for the treatment of disease MAP3K20, MAP3K1, MAP3K2 NPC1 1115/4885ALDH1A1 3678/4885RAB9A 3067/4885
US-20030187007-A1 Inhibitors of protein kinase for the treatment of disease MAP3K20, MAP3K1, MAP3K2 NPC1 1115/4885ALDH1A1 3678/4885RAB9A 3067/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.