SCHEMBL6646707

SCHEMBL6646707

O=c1[nH]c(CCCC2CC(c3ccccc3)=CCN2)nc2c1CCC2

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.58
HTR1A P08908 1/20 0.42
HTR3A P46098 1/20 0.42
PKM P14618 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HPGD P15428 4/20 0.40
HTR2C P28335 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 2/20 0.37
ALPL P05186 1/20 0.37
ALPI P09923 1/20 0.37
ALPG P10696 1/20 0.37
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6648890 0.98 PARP1 (0.56) PARP1HTR1AHTR3APKML3MBTL1
SCHEMBL6651055 0.87 PARP1 (0.45) PARP1HTR1AHTR3AHTR2CTNKS
SCHEMBL6649328 0.86 PARP1 (0.44) PARP1HTR1AHTR3AHTR2CTNKS
SCHEMBL6418477 0.85 PARP1 (0.43) PARP1HTR2CTNKSTNKS2
SCHEMBL6650044 0.85 PARP1 (0.51) PARP1HTR1AHTR3A
Hydrochloric Acid SCHEMBL7018458 0.81 PARP1 (0.55) PARP1
SCHEMBL7023192 0.78 PARP1 (0.49) PARP1
SCHEMBL467535 0.77 PARP1 (0.60) PARP1
SCHEMBL7017894 0.77 PARP1 (0.48) PARP1
SCHEMBL7017660 0.77 PARP1 (0.60) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1469854-A1 CONDENSED HETEROCYCLIC COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-10-27 EP disclosed
WO-2003063874-A1 CONDENSED HETEROCYCLIC COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-08-07 WO disclosed