SCHEMBL6650044

SCHEMBL6650044

CN1CCc2nc(CCCC3CC(c4ccccc4)=CCN3)[nH]c(=O)c2C1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.51
HTR1A P08908 1/20 0.37
HTR3A P46098 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6648890 0.85 PARP1 (0.56) PARP1HTR1AHTR3A
SCHEMBL6646707 0.85 PARP1 (0.58) PARP1HTR1AHTR3A
SCHEMBL6651055 0.82 PARP1 (0.45) PARP1HTR1AHTR3A
SCHEMBL6649328 0.81 PARP1 (0.44) PARP1HTR1AHTR3A
SCHEMBL6418477 0.80 PARP1 (0.43) PARP1
SCHEMBL7016636 0.79 PARP1 (0.51) PARP1HTR1A
SCHEMBL6368822 0.79 PARP1 (0.77) PARP1
Hydrochloric Acid SCHEMBL7018458 0.77 PARP1 (0.55) PARP1
SCHEMBL6651964 0.74 PARP1 (0.42) PARP1
SCHEMBL7023192 0.74 PARP1 (0.49) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1469854-A1 CONDENSED HETEROCYCLIC COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-10-27 EP disclosed
WO-2003063874-A1 CONDENSED HETEROCYCLIC COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-08-07 WO disclosed