SCHEMBL6648928

SCHEMBL6648928

COc1cccc(CNC(Cc2cc(F)cc(F)c2)C(O)CNC(=O)c2cc(C)cc(C(O)c3ccccc3C)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.54
BACE2 Q9Y5Z0 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3351517 0.89 BACE1 (0.69) BACE1BACE2
SCHEMBL3351524 0.89 BACE1 (0.69) BACE1BACE2
SCHEMBL6893064 0.81 BACE1 (0.54) BACE1BACE2
SCHEMBL3346953 0.75 BACE1 (0.72) BACE1BACE2
SCHEMBL3346959 0.75 BACE1 (0.72) BACE1BACE2
SCHEMBL3355738 0.75 BACE1 (0.77) BACE1BACE2
SCHEMBL3355743 0.75 BACE1 (0.77) BACE1BACE2
SCHEMBL5121674 0.75 BACE1 (0.47) BACE1BACE2
SCHEMBL5350790 0.74 BACE1 (0.79) BACE1BACE2
SCHEMBL16578190 0.74 BACE1 (0.91) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453789-A2 N,N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES Elan Pharmaceuticals, Inc. (US) 2004-09-08 EP claimed
WO-2003040096-A2 N, N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES ELAN PHARMACEUTICALS, INC. (US) 2003-05-15 WO claimed