SCHEMBL6650864

SCHEMBL6650864

CC(=O)c1c(C)nc2ccccc2c1NCc1ccc(Br)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.51
HSD17B10 Q99714 1/20 0.51
APP P05067 4/20 0.51
ALDH1A1 P00352 2/20 0.49
KMT2A Q03164 2/20 0.49
POLB P06746 2/20 0.49
RAD52 P43351 1/20 0.49
HTT P42858 2/20 0.47
NTRK1 P04629 1/20 0.44
ACHE P22303 1/20 0.44
MEN1 O00255 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PRNP P04156 1/20 0.42
PPARG P37231 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
NR2E3 Q9Y5X4 1/20 0.42
NCOR2 Q9Y618 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653573 0.92 APP (0.52) TP53HSD17B10APPALDH1A1KMT2A
SCHEMBL9821131 0.91 KMT2A (0.59) TP53HSD17B10APPALDH1A1KMT2A
Hydrochloric Acid SCHEMBL9821072 0.90 KMT2A (0.57) TP53HSD17B10APPALDH1A1KMT2A
SCHEMBL7649849 0.88 KMT2A (0.55) TP53APPALDH1A1KMT2APOLB
SCHEMBL9821213 0.88 HTT (0.52) TP53HSD17B10APPALDH1A1KMT2A
SCHEMBL6658584 0.88 HSD17B10 (0.51) TP53HSD17B10APPALDH1A1KMT2A
SCHEMBL7649838 0.87 APP (0.54) TP53HSD17B10APPALDH1A1KMT2A
Hydrochloric Acid SCHEMBL10567928 0.87 KMT2A (0.53) TP53HSD17B10APPALDH1A1KMT2A
SCHEMBL6657077 0.85 TP53 (0.45) TP53HSD17B10APPALDH1A1KMT2A
SCHEMBL7647477 0.85 TP53 (0.45) TP53HSD17B10APPALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218401-B1 4-BENZYLAMINOQUINOLINE CONJUGATES WITH BILE ACID AND THEIR HETEROANALOGUES, METHODS FOR PRODUCING THE SAME, MEDICAMENTS CONTAINING THESE COMPOUNDS AND THEIR USE AVENTIS PHARMA GMBH (DE) 2004-06-16 EP disclosed
EP-1218401-A1 4-BENZYLAMINOQUINOLINE CONJUGATES WITH BILE ACID AND THEIR HETEROANALOGUES, METHODS FOR PRODUCING THE SAME, MEDICAMENTS CONTAINING THESE COMPOUNDS AND THEIR USE Aventis Pharma Deutschland GmbH (DE) 2002-07-03 EP disclosed
US-6339077-B1 FOR PROPHYLAXIS OR OF GALLSTONES AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-01-15 US disclosed
WO-2001021642-A1 4-BENZYLAMINOQUINOLINE CONJUGATES WITH BILE ACID AND THEIR HETEROANALOGUES, METHODS FOR PRODUCING THE SAME, MEDICAMENTS CONTAINING THESE COMPOUNDS AND THEIR USE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-03-29 WO disclosed