SCHEMBL6651828

SCHEMBL6651828

c1ccc2c(CC3NCCc4c3[nH]c3ccccc43)cccc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 8/20 0.69
CHRM4 P08173 5/20 0.69
GRIN2B Q13224 1/20 0.68
CTSK P43235 1/20 0.59
DRD2 P14416 3/20 0.58
CYP2D6 P10635 2/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C19 P33261 1/20 0.52
HTR2A P28223 3/20 0.51
HTR2C P28335 1/20 0.51
ALDH1A1 P00352 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9393283 0.99 HTR7 (0.68) HTR7CHRM4GRIN2BCTSKDRD2
SCHEMBL8683890 0.87 HTR7 (0.55) HTR7CHRM4GRIN2BCTSKDRD2
Hydrochloric Acid SCHEMBL8684071 0.86 HTR2B (0.58) HTR7CHRM4GRIN2BDRD2HTR2A
Hydrochloric Acid SCHEMBL8684280 0.86 HTR2B (0.58) HTR7CHRM4GRIN2BDRD2HTR2A
SCHEMBL8906099 0.86 HTR7 (0.64) HTR7CHRM4GRIN2BCTSKDRD2
Hydrochloric Acid SCHEMBL8938691 0.85 HTR2A (0.56) HTR7CHRM4GRIN2BDRD2HTR2A
SCHEMBL8685840 0.85 HTR7 (0.52) HTR7CHRM4GRIN2BCTSKDRD2
SCHEMBL8907199 0.85 HTR7 (0.63) HTR7CHRM4GRIN2BCTSKDRD2
Hydrochloric Acid SCHEMBL7818446 0.85 HTR7 (0.54) HTR7CHRM4GRIN2BCTSKDRD2
SCHEMBL8938572 0.85 HTR7 (0.54) HTR7CHRM4GRIN2BDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389194-A2 INHIBITORS OF BACE VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-02-18 EP disclosed
WO-2002088101-A2 INHIBITORS OF BACE VERTEX PHARMACEUTICALS INCORPORATED (US) 2002-11-07 WO disclosed