SCHEMBL6651987

SCHEMBL6651987

COC(=O)c1ccc(C2=CCCCC2)c(C)c1.Cc1cc(C(=O)O)ccc1C1=CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.42
ALDH1A1 P00352 5/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
KDM6B O15054 1/20 0.41
KDM5C P41229 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM2A Q9Y2K7 1/20 0.41
KDM3A Q9Y4C1 1/20 0.41
GAA P10253 2/20 0.40
ACMSD Q8TDX5 1/20 0.39
MAPT P10636 2/20 0.38
CLCN2 P51788 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
ATM Q13315 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6068829 0.95 CA12 (0.41) KDM4EALDH1A1MEN1KMT2ANPC1
SCHEMBL4950570 0.91 CA12 (0.41) KDM4EALDH1A1NPC1RAB9AGAA
SCHEMBL6068947 0.91 GAA (0.45) KDM4EALDH1A1MEN1KMT2ANPC1
SCHEMBL28268790 0.81 KDM4E (0.54) KDM4EALDH1A1MEN1KMT2AKDM6B
SCHEMBL24834901 0.81 GRM2 (0.41) KDM4EALDH1A1MEN1KMT2ANPC1
SCHEMBL3904050 0.80 NOTUM (0.49) KDM4EALDH1A1MEN1KMT2ANPC1
SCHEMBL2501250 0.78 CA12 (0.50) KDM4EALDH1A1MEN1KMT2ANPC1
SCHEMBL6632862 0.77 SMN1; SMN2 (0.38) KDM4EALDH1A1MEN1KMT2ANPC1
SCHEMBL22077172 0.76 NOTUM (0.50) KDM4EALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL27902795 0.76 ACMSD (0.52) KDM4EALDH1A1GAAACMSDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377584-A1 NOVEL CYCLOHEXENYL PHENYL DIAZEPINES AS VASOPRESSIN AND OXYTOCIN RECEPTOR MODULATORS Wyeth (US) 2004-01-07 EP disclosed
WO-2002083681-A1 NOVEL CYCLOHEXENYL PHENYL DIAZEPINES VASOPRESSIN AND OXYTOCIN RECEPTOR MODULATORS WYETH (US) 2002-10-24 WO disclosed