SCHEMBL6651993

SCHEMBL6651993

Cc1ccncc1-c1nc(-c2ccccc2Cl)cs1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.59
L3MBTL1 Q9Y468 3/20 0.56
LMNA P02545 2/20 0.56
KMT2A Q03164 2/20 0.56
MAPT P10636 1/20 0.56
RAB9A P51151 4/20 0.51
NPC1 O15118 3/20 0.51
KDM4E B2RXH2 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
C1S P09871 1/20 0.47
CYP1A2 P05177 3/20 0.46
CYP1A1 P04798 2/20 0.46
CYP1B1 Q16678 2/20 0.46
ALDH1A1 P00352 3/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
CYP17A1 P05093 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
ATP4A P20648 2/20 0.44
ATP4B P51164 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3818666 0.85 CYP19A1 (0.55) CYP19A1L3MBTL1LMNAKMT2AMAPT
SCHEMBL6626985 0.84 SMN1; SMN2 (0.51) CYP19A1LMNAKMT2AMAPTRAB9A
SCHEMBL6648194 0.83 RAB9A (0.65) CYP19A1L3MBTL1LMNAKMT2AMAPT
SCHEMBL6648164 0.83 CYP19A1 (0.56) CYP19A1L3MBTL1LMNAKMT2AMAPT
Hydrochloric Acid SCHEMBL6627345 0.83 SMN1; SMN2 (0.50) CYP19A1LMNAKMT2AMAPTRAB9A
SCHEMBL6651305 0.83 CYP19A1 (0.56) CYP19A1L3MBTL1LMNAKMT2AMAPT
SCHEMBL6646978 0.82 CYP19A1 (0.58) CYP19A1L3MBTL1LMNAKMT2AMAPT
SCHEMBL6648550 0.82 RAB9A (0.63) CYP19A1L3MBTL1LMNAKMT2AMAPT
SCHEMBL6648165 0.81 CYP19A1 (0.53) CYP19A1L3MBTL1LMNAKMT2AMAPT
SCHEMBL3821580 0.79 KDM4E (0.61) CYP19A1LMNAKMT2ARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432706-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
WO-2003027085-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed