SCHEMBL6653668

SCHEMBL6653668

CCCCCc1ccc(C(=O)c2ccc(N)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RARB P10826 5/20 0.58
THRA P10827 9/20 0.57
THRB P10828 9/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
ALDH1A1 P00352 2/20 0.57
RARA P10276 1/20 0.57
MAPT P10636 1/20 0.57
MTOR P42345 1/20 0.57
HTR2A P28223 1/20 0.55
PLA2G1B P04054 2/20 0.54
ATG4B Q9Y4P1 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11086601 0.98 THRA (0.59) RARBTHRATHRBMEN1KMT2A
SCHEMBL11202747 0.98 THRA (0.59) RARBTHRATHRBMEN1KMT2A
SCHEMBL10580743 0.95 RARB (0.57) RARBTHRATHRBMEN1KMT2A
SCHEMBL617127 0.91 RARB (0.68) RARBTHRATHRBMEN1KMT2A
SCHEMBL16536411 0.89 THRA (0.69) RARBTHRATHRBMEN1KMT2A
SCHEMBL7652503 0.89 THRA (0.69) RARBTHRATHRBMEN1KMT2A
SCHEMBL15453509 0.89 THRA (0.69) RARBTHRATHRBMEN1KMT2A
SCHEMBL7649277 0.89 THRA (0.69) RARBTHRATHRBMEN1KMT2A
SCHEMBL2970920 0.89 THRA (0.69) RARBTHRATHRBMEN1KMT2A
SCHEMBL28963426 0.89 THRA (0.69) RARBTHRATHRBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966424-B1 AMINOBENZOPHENONES AS INHIBITORS OF INTERLEUKIN AND TNF LEO PHARMA AS (DK) 2004-06-23 EP disclosed
US-6313174-B1 FOR THERAPY AND PROPHYLAXIS OF ASTHMA, ALLERGY, RHEUMATOID ARTHRITIS, SPONDYLOARTHRITIS, GOUT, ATHEROSCLEROSIS, CHRONIC INFLAMMATORY BOWEL DISEASE, PROLIFERATIVE AND INFLAMMATORY SKIN DISORDERS Leo Pharmaceutical Products Ltd.A/S/ (Løvens kemiske Fabrik Produktionsaktieselskab) (DK) 2001-11-06 US disclosed
EP-0966424-A1 AMINOBENZOPHENONES AS INHIBITORS OF INTERLEUKIN AND TNF LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 1999-12-29 EP disclosed
WO-1998032730-A1 AMINOBENZOPHENONES AS INHIBITORS OF INTERLEUKIN AND TNF Leo Pharmaceutical Products Ltd. A/S (Løvens Kemiske Fabrik Produktionsaktieselskab) (DK) 1998-07-30 WO disclosed
EP-0302401-A1 Pyridone dyes, process for their preparation and their use CASSELLA Aktiengesellschaft (DE) 1989-02-08 EP disclosed