SCHEMBL6654411

SCHEMBL6654411

CCCc1ccncc1-c1nc(-c2cccc(Cl)c2)cs1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.55
MAPT P10636 3/20 0.48
GLA P06280 1/20 0.48
SREBF2 Q12772 4/20 0.47
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
ATM Q13315 1/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP1B1 Q16678 1/20 0.43
LIMK1 P53667 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6646768 0.92 CYP19A1 (0.56) CYP19A1MAPTGLANPC1RAB9A
SCHEMBL6646066 0.86 RAB9A (0.48) CYP19A1MAPTSREBF2KDM4ELMNA
SCHEMBL6648190 0.86 KDM4E (0.52) CYP19A1MAPTSREBF2KDM4ENPC1
SCHEMBL6647164 0.85 KDM4E (0.59) CYP19A1MAPTSREBF2KDM4ELMNA
SCHEMBL6646344 0.85 KDM4E (0.57) CYP19A1SREBF2KDM4ENPC1RAB9A
SCHEMBL6650025 0.84 C1S (0.47) CYP19A1MAPTSREBF2KDM4ELMNA
SCHEMBL6648508 0.84 KDM4E (0.51) CYP19A1MAPTSREBF2KDM4ELMNA
SCHEMBL6646582 0.83 CYP19A1 (0.60) CYP19A1MAPTGLAKDM4ELMNA
SCHEMBL6650443 0.83 SREBF2 (0.55) CYP19A1SREBF2KDM4ENPC1RAB9A
SCHEMBL6649816 0.82 CDC25A (0.55) CYP19A1MAPTSREBF2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432706-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
WO-2003027085-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed