SCHEMBL6655

SCHEMBL6655

COc1ccc(C(C)CCNc2c(C)noc2-c2ccc(Br)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
L3MBTL1 Q9Y468 2/20 0.38
HTT P42858 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
LPAR1 Q92633 3/20 0.38
LPAR3 Q9UBY5 1/20 0.38
ALDH1A1 P00352 3/20 0.36
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
RAB9A P51151 2/20 0.34
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
LMNA P02545 2/20 0.33
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7648 0.89 MEN1 (0.44) MEN1KMT2AL3MBTL1HTTTDP1
SCHEMBL2106 0.87 MAPT (0.39) LPAR1LPAR3EDNRBEDNRAMAPT
SCHEMBL1166 0.87 LPAR1 (0.47) LPAR1LPAR3ALDH1A1EDNRBEDNRA
SCHEMBL1651 0.79 LPAR1 (0.39) LPAR1LPAR3ALDH1A1EDNRBEDNRA
SCHEMBL1579 0.79 LPAR1 (0.39) LPAR1LPAR3ALDH1A1LMNAABCC3
SCHEMBL2096 0.77 MAPT (0.46) MEN1KMT2AL3MBTL1HTTTDP1
SCHEMBL6665 0.77 MEN1 (0.45) MEN1KMT2AL3MBTL1HTTTDP1
SCHEMBL1733 0.77 LPAR1 (0.37) LPAR1LPAR3MAPTGAANPSR1
SCHEMBL2195 0.77 LPAR1 (0.48) MEN1KMT2AHTTTDP1LPAR1
SCHEMBL343959 0.76 LPAR1 (0.68) MEN1KMT2ALPAR1LPAR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed