SCHEMBL6656526

SCHEMBL6656526

Cc1[nH]c2ccc(O)cc2c1C(=O)OCc1ccccc1.Cc1[nH]c2ccc(OCCCBr)cc2c1C(=O)OCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.56
ALOX5 P09917 7/20 0.51
KMT2A Q03164 2/20 0.49
KDM4E B2RXH2 2/20 0.49
LMNA P02545 2/20 0.49
MAPT P10636 2/20 0.49
HPGD P15428 2/20 0.49
HSD17B10 Q99714 2/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPK10 P53779 1/20 0.49
GABRA1 P14867 2/20 0.46
GABRG2 P18507 2/20 0.46
GABRB3 P28472 2/20 0.46
GABRA5 P31644 2/20 0.46
GABRA3 P34903 2/20 0.46
GABRA2 P47869 2/20 0.46
TRPM8 Q7Z2W7 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6315741 0.96 GAA (0.49) GAAALOX5KMT2AKDM4ELMNA
SCHEMBL6315808 0.87 GAA (0.74) GAAALOX5KMT2AKDM4ELMNA
SCHEMBL6317769 0.86 GAA (0.49) GAAALOX5KMT2AKDM4ELMNA
SCHEMBL6314661 0.85 GAA (0.50) GAAALOX5KMT2AKDM4ELMNA
SCHEMBL6316345 0.85 GAA (0.50) GAAALOX5KMT2AKDM4ELMNA
SCHEMBL6321136 0.83 GAA (0.54) GAAALOX5KMT2AKDM4ELMNA
SCHEMBL6315202 0.83 GAA (0.48) GAAALOX5KMT2AKDM4ELMNA
SCHEMBL6656803 0.82 GAA (0.57) GAAALOX5KMT2AKDM4ELMNA
SCHEMBL6314855 0.81 NPC1 (0.54) KDM4EALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL6654441 0.81 GAA (0.46) GAAALOX5KMT2AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377549-A1 FUNCTIONALIZED HETEROCYCLES AS MODULATORS OF CHEMOKINE RECEPTOR FUNCTION AND METHODS OF USE THEREFOR Millennium Pharmaceuticals, Inc. (US) 2004-01-07 EP disclosed
WO-2002072549-A1 FUNCTIONALIZED HETEROCYCLES AS MODULATORS OF CHEMOKINE RECEPTOR FUNCTION AND METHODS OF USE THEREFOR MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-09-19 WO disclosed