SCHEMBL6657766

SCHEMBL6657766

NC(Cc1ccncc1)C(=O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 16/20 0.59
ROCK2 O75116 1/20 0.52
CYP3A4 P08684 1/20 0.52
AKT2 P31751 7/20 0.50
AKT3 Q9Y243 7/20 0.50
CHRM1 P11229 1/20 0.48
HRH2 P25021 2/20 0.48
HRH1 P35367 2/20 0.48
AKT1S1 Q96B36 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6657763 1.00 AKT1 (0.59) AKT1ROCK2CYP3A4AKT2AKT3
Hydrochloric Acid SCHEMBL3960080 0.99 AKT1 (0.58) AKT1ROCK2CYP3A4AKT2AKT3
SCHEMBL7010740 0.86 AKT1 (0.49) AKT1ROCK2CYP3A4AKT2AKT3
SCHEMBL4213022 0.85 AKT1 (0.54) AKT1AKT2AKT3CHRM1HRH2
SCHEMBL4213020 0.85 AKT1 (0.54) AKT1AKT2AKT3CHRM1HRH2
SCHEMBL10180336 0.85 AKT1 (0.54) AKT1AKT2AKT3CHRM1HRH2
SCHEMBL3954177 0.85 CALCRL (0.53) AKT1ROCK2CYP3A4AKT2AKT3
SCHEMBL6268215 0.84 AKT1 (0.51) AKT1CHRM1HRH2HRH1
SCHEMBL7005623 0.84 AKT1 (0.47) AKT1ROCK2CYP3A4AKT2AKT3
SCHEMBL7005621 0.84 AKT1 (0.47) AKT1ROCK2CYP3A4AKT2AKT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440976-A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production Boehringer Ingelheim Pharma GmbH & Co.KG (DE) 2004-07-28 EP disclosed