SCHEMBL7010740

SCHEMBL7010740

N[C@H](Cc1cc(Br)c(O)c(Br)c1)C(=O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 4/20 0.49
CALCRL Q16602 15/20 0.48
ROCK2 O75116 1/20 0.46
CYP3A4 P08684 1/20 0.46
RAMP1 O60894 5/20 0.46
AKT2 P31751 1/20 0.44
AKT3 Q9Y243 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3954177 0.92 CALCRL (0.53) AKT1CALCRLROCK2CYP3A4RAMP1
SCHEMBL7005623 0.91 AKT1 (0.47) AKT1CALCRLROCK2CYP3A4RAMP1
SCHEMBL7005621 0.91 AKT1 (0.47) AKT1CALCRLROCK2CYP3A4RAMP1
SCHEMBL5618860 0.88 AKT1 (0.53) AKT1CALCRLROCK2CYP3A4RAMP1
SCHEMBL6657766 0.86 AKT1 (0.59) AKT1ROCK2CYP3A4AKT2AKT3
SCHEMBL6657763 0.86 AKT1 (0.59) AKT1ROCK2CYP3A4AKT2AKT3
SCHEMBL4717217 0.86 AKT1 (0.48) AKT1CALCRLROCK2CYP3A4AKT2
Hydrochloric Acid SCHEMBL3960080 0.85 AKT1 (0.58) AKT1ROCK2CYP3A4AKT2AKT3
SCHEMBL3964152 0.83 SMYD3 (0.49) AKT1CALCRLROCK2CYP3A4RAMP1
SCHEMBL18822516 0.79 CALCRL (0.64) CALCRLRAMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163239-B1 MODIFIED AMINO-ACID AMIDES AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM PHARMA (DE) 2003-05-28 EP disclosed
US-6313097-B1 TREATMENT OR PROPHYLAXIS OF MIGRAINE OR CLUSTER HEADACHES, NON-INSULIN-DEPENDENT DIABETES MELLITUS, INFLAMMATION, ALLERGIC RHINITIS, ASTHMA, MORPHINE TOLERANCE, MENOPAUSAL HOT FLASHES, DISEASES CHARACTERIZED BY EXCESSIVE VASODILATATION BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-11-06 US disclosed