⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL29086344 | 0.85 | CYP1B1 (0.32) | — | |
| SCHEMBL14764836 | 0.83 | HDAC3 (0.34) | — | |
| SCHEMBL125617 | 0.80 | — | — | |
| SCHEMBL7022926 | 0.78 | FAAH (0.38) | — | |
| SCHEMBL7029638 | 0.78 | FAAH (0.38) | — | |
| SCHEMBL7027055 | 0.78 | FAAH (0.38) | — | |
| SCHEMBL1680363 | 0.78 | — | — | |
| SCHEMBL20813055 | 0.77 | — | — | |
| SCHEMBL6410587 | 0.77 | — | — | |
| SCHEMBL6012846 | 0.76 | — | — |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 146 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-2032124-A1 | MULTIPARTICULATE OSMOTIC DELIVERY SYSTEM | BIOVAIL LABORATORIES INTERNATIONAL SRL (BB) | 2009-03-11 | — | — | EP | claimed |
| US-20090004281-A1 | MULTIPARTICULATE OSMOTIC DELIVERY SYSTEM | BIOVAIL LABORATORIES INTERNATIONAL S.R.L. (BB) | 2009-01-01 | — | — | US | claimed |
| WO-2008001341-A1 | MULTIPARTICULATE OSMOTIC DELIVERY SYSTEM | BIOVAIL LABORATORIES INTERNATIONAL SRL (BB) | 2008-01-03 | — | — | WO | claimed |
| US-20050182022-A1 | Chondroprotective/restorative compositions and methods of use thereof | PIERCE SCOTT W (US) | 2005-08-18 | — | — | US | claimed |
| US-6924273-B2 | Chondroprotective/restorative compositions and methods of use thereof | PIERCE SCOTT W (US) | 2005-08-02 | — | — | US | claimed |
| EP-0746342-B1 | BIODEGRADABLE CONTROLLED RELEASE MELT-SPUN DELIVERY SYSTEM | BIOVAIL TECH LTD (US) | 2002-08-14 | — | — | EP | claimed |
| US-20020068718-A1 | Chondroprotective/restorative compositions and methods of use thereof | PIERCE SCOTT W (US) | 2002-06-06 | — | — | US | claimed |
| EP-0746342-A1 | BIODEGRADABLE CONTROLLED RELEASE MELT-SPUN DELIVERY SYSTEM | FUISZ TECHNOLOGIES LTD. (US) | 1996-12-11 | — | — | EP | claimed |
| US-5518730-A | Biodegradable controlled release flash flow melt-spun delivery system | FUISZ TECHNOLOGIES LTD. (US) | 1996-05-21 | — | — | US | claimed |
| EP-0746342-A4 | BIODEGRADABLE CONTROLLED RELEASE MELT-SPUN DELIVERY SYSTEM | FUISZ TECHNOLOGIES LTD (US) | 1996-01-11 | — | — | EP | claimed |
| WO-1993024154-A1 | BIODEGRADABLE CONTROLLED RELEASE MELT-SPUN DELIVERY SYSTEM | FUISZ TECHNOLOGIES, LTD. (US) | 1993-12-09 | — | — | WO | claimed |
| US-11091464-B2 | Pyridazinone compounds and uses thereof | EDGEWISE THERAPEUTICS, INC. (US) | 2021-08-17 | — | — | US | disclosed |
| US-9549767-B2 | Encapsulated screw locking system | STRYKER EUROPEAN HOLDINGS I, LLC (US) | 2017-01-24 | — | — | US | disclosed |
| US-9050264-B2 | Cellulose capsules and methods for making them | UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) | 2015-06-09 | — | — | US | disclosed |
| EP-2335628-B1 | Therapeutic agent capsule for implants | STRYKER TRAUMA GMBH (DE) | 2013-11-27 | — | — | EP | disclosed |
| EP-0746342-A1 | BIODEGRADABLE CONTROLLED RELEASE MELT-SPUN DELIVERY SYSTEM | FUISZ TECHNOLOGIES LTD. (US) | 1996-12-11 | — | — | EP | disclosed |
| US-5518730-A | Biodegradable controlled release flash flow melt-spun delivery system | FUISZ TECHNOLOGIES LTD. (US) | 1996-05-21 | — | — | US | disclosed |
| EP-0746342-A4 | BIODEGRADABLE CONTROLLED RELEASE MELT-SPUN DELIVERY SYSTEM | FUISZ TECHNOLOGIES LTD (US) | 1996-01-11 | — | — | EP | disclosed |
| WO-1993024154-A1 | BIODEGRADABLE CONTROLLED RELEASE MELT-SPUN DELIVERY SYSTEM | FUISZ TECHNOLOGIES, LTD. (US) | 1993-12-09 | — | — | WO | disclosed |
| WO-1992015285-A1 | STARCH-BASED CONTROLLED RELEASE COMPOSITIONS | WARNER-LAMBERT COMPANY (US) | 1992-09-17 | — | — | WO | disclosed |