SCHEMBL6658034

SCHEMBL6658034

O=C(NCc1cccc(O)c1)c1cc2ccccc2[nH]1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.81
CA12 O43570 1/20 0.61
CA1 P00915 1/20 0.61
CA2 P00918 1/20 0.61
CA9 Q16790 1/20 0.61
IDO1 P14902 2/20 0.59
OPRK1 P41145 1/20 0.59
HDAC2 Q92769 2/20 0.58
HDAC3 O15379 1/20 0.58
HDAC1 Q13547 1/20 0.58
NCOR2 Q9Y618 1/20 0.58
KDM4E B2RXH2 4/20 0.57
ALDH1A1 P00352 2/20 0.57
GAA P10253 1/20 0.57
MAPK1 P28482 1/20 0.57
DRD2 P14416 1/20 0.55
DRD3 P35462 1/20 0.55
HSD17B10 Q99714 1/20 0.55
MIF P14174 1/20 0.55
AKR1C3 P42330 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2735957 0.90 SRC (1.00) SRCCA12CA1CA2CA9
SCHEMBL2735969 0.88 CA12 (0.72) SRCCA12CA1CA2CA9
SCHEMBL6657027 0.86 HDAC2 (0.67) SRCCA12CA1CA2CA9
SCHEMBL17149769 0.86 LMNA (0.62) SRCCA12CA1CA2CA9
SCHEMBL2735774 0.85 SRC (0.82) SRCCA12CA1CA2CA9
SCHEMBL29381586 0.85 SRC (0.82) SRCCA12CA1CA2CA9
SCHEMBL12763661 0.85 SRC (0.82) SRCCA12CA1CA2CA9
SCHEMBL2760003 0.83 SRC (0.83) SRCCA12CA1CA2CA9
SCHEMBL6300914 0.81 HDAC2 (0.57) SRCCA12CA1CA2CA9
SCHEMBL12763659 0.80 SRC (0.82) SRCCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440966-A1 Indole derivatives useful for the treatment of diseases Pfizer Limited (GB) 2004-07-28 EP disclosed