SCHEMBL6659477

SCHEMBL6659477

CC(=O)Nc1ccc(-c2c3c(=O)n(C)c(=O)n(CC(C)C)c3nn2Cc2ccccc2-c2ccc(F)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.41
MAPT P10636 2/20 0.41
PDE1A P54750 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE1C Q14123 1/20 0.39
ADORA2B P29275 2/20 0.38
ADORA1 P30542 2/20 0.38
THRB P10828 1/20 0.38
KCNA5 P22460 1/20 0.37
KCNH2 Q12809 1/20 0.37
LMNA P02545 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HSD17B10 Q99714 1/20 0.37
DPP4 P27487 1/20 0.36
PDE5A O76074 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5404652 0.87 RIPK3 (0.41) PDE1APDE1BPDE1CLMNAPDE5A
SCHEMBL5405288 0.86 SLC16A1 (0.47) TP53MAPTPDE1APDE1BPDE1C
SCHEMBL5407653 0.84 TP53 (0.40) TP53MAPTPDE1APDE1BPDE1C
SCHEMBL5400727 0.84 TP53 (0.39) TP53MAPTPDE1APDE1BPDE1C
SCHEMBL5417969 0.84 MEN1 (0.39) PDE1APDE1BPDE1CADORA2BKCNA5
SCHEMBL5405558 0.83 SLC16A1 (0.47) TP53MAPTPDE1APDE1BPDE1C
SCHEMBL5399340 0.82 PDE5A (0.37) PDE1APDE1BPDE1CLMNAPDE5A
SCHEMBL5405716 0.82 TP53 (0.44) TP53MAPTPDE1APDE1BPDE1C
SCHEMBL5404004 0.81 MAPT (0.40) TP53MAPTPDE1APDE1BPDE1C
SCHEMBL5399832 0.81 PDE5A (0.37) PDE1APDE1BPDE1CPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1412355-A1 NEW PYRAZOLO(3,4-D)PYRIMIDINES INHIBITING H. PYLORI INFECTIONS AstraZeneca AB (SE) 2004-04-28 EP disclosed
WO-2003002567-A1 NEW PYRAZOLO[3,4-D]PYRIMIDINES INHIBITING H. PYLORI INFECTIONS ASTRAZENECA AB (SE) 2003-01-09 WO disclosed