SCHEMBL6659650

SCHEMBL6659650

CSc1ccc(-c2nc3c(Cl)ncnc3n2C2CCCCO2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.38
ADORA3 P0DMS8 10/20 0.37
ADORA2A P29274 10/20 0.37
ADORA1 P30542 10/20 0.37
YTHDC1 Q96MU7 1/20 0.36
ADORA2B P29275 5/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TP53 P04637 1/20 0.33
CYP2C9 P11712 1/20 0.33
NFKB1 P19838 1/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
APEX1 P27695 1/20 0.33
PI4KA P42356 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29877869 0.80 CYP2C19 (0.45) CYP1A2TSHRCYP2C19ADORA3ADORA2A
SCHEMBL14964663 0.80 CYP2C19 (0.45) CYP1A2TSHRCYP2C19ADORA3ADORA2A
SCHEMBL17847271 0.77 PI4KA (0.46) CYP1A2TSHRCYP2C19ADORA3ADORA2A
SCHEMBL12068396 0.77 CYP2C19 (0.43) CYP1A2TSHRCYP2C19ADORA3ADORA2A
SCHEMBL5724445 0.77 CYP1A2 (0.50) CYP1A2TSHRCYP2C19ADORA3ADORA2A
SCHEMBL783034 0.76 CYP1A2 (0.40) CYP1A2TSHRCYP2C19ADORA3ADORA2A
SCHEMBL6664608 0.76 ADORA3 (0.47) CYP1A2TSHRCYP2C19ADORA3ADORA2A
SCHEMBL29877816 0.75 CYP2C19 (0.43) CYP1A2TSHRCYP2C19ADORA3ADORA2A
SCHEMBL6659013 0.74 ADORA3 (0.48) ADORA3ADORA2AADORA1ADORA2BALDH1A1
SCHEMBL21685107 0.73 CYP1A2 (0.44) CYP1A2TSHRCYP2C19ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444982-A1 The use of purine derivatives as selective kinase inhibitors MERCKLE GMBH (DE) 2004-08-11 EP disclosed