SCHEMBL6662884

SCHEMBL6662884

NC(=O)CC(Cc1ccc(Cl)cc1)c1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 6/20 0.51
GABBR1 Q9UBS5 6/20 0.51
CYP2C9 P11712 3/20 0.51
LMNA P02545 3/20 0.51
CYP2C19 P33261 2/20 0.51
CYP1A2 P05177 2/20 0.51
THRB P10828 2/20 0.51
CYP3A4 P08684 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
NFKB1 P19838 1/20 0.51
DRD3 P35462 1/20 0.51
BLM P54132 1/20 0.51
CYP2D6 P10635 1/20 0.51
MEN1 O00255 1/20 0.51
TSHR P16473 1/20 0.51
KMT2A Q03164 1/20 0.51
SLC6A4 P31645 1/20 0.46
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL523877 0.87 GABBR2 (0.59) GABBR2GABBR1CYP2C9LMNACYP2C19
SCHEMBL5273737 0.83 GABBR2 (0.42) GABBR2GABBR1
SCHEMBL7031963 0.82 GABBR2 (0.74) GABBR2GABBR1CYP2C9LMNACYP2C19
SCHEMBL22172484 0.81 GABBR2 (0.72) GABBR2GABBR1CYP2C9LMNACYP2C19
SCHEMBL12883209 0.81 GABBR2 (0.53) GABBR2GABBR1CYP2C9LMNACYP2C19
SCHEMBL7822991 0.81 GABBR2 (0.72) GABBR2GABBR1CYP2C9LMNACYP2C19
SCHEMBL5801572 0.79 EPHX1 (0.58) GABBR2GABBR1CYP2C19CYP1A2CYP2D6
SCHEMBL11298234 0.79 SLC6A4 (0.48) CYP2C9CYP2C19CYP1A2CYP2D6SLC6A4
SCHEMBL16439493 0.78 GABBR2 (0.58) GABBR2GABBR1CYP2C9LMNACYP2C19
Hydrochloric Acid SCHEMBL7314689 0.77 EPHX1 (0.56) GABBR2GABBR1CYP2C19CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004103278-A2 ACYL SULFONAMIDES AS INHIBITORS OF HIV INTEGRASE BRISTOL-MYERS SQUIBB COMPANY (US) 2004-12-02 WO claimed
WO-2004103278-A2 ACYL SULFONAMIDES AS INHIBITORS OF HIV INTEGRASE BRISTOL-MYERS SQUIBB COMPANY (US) 2004-12-02 WO disclosed
WO-2004004657-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-01-15 WO disclosed