SCHEMBL6663541

SCHEMBL6663541

NC(=O)c1nn(-c2ccc(S(N)(=O)=O)cc2)c2c1CCc1cnccc1-2

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 16/20 0.65
CDK2 P24941 16/20 0.65
CCNA1 P78396 16/20 0.65
IKBKB O14920 1/20 0.65
AURKA O14965 2/20 0.55
PTGS1 P23219 2/20 0.51
PTGS2 P35354 2/20 0.51
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA4 P22748 2/20 0.45
CA9 Q16790 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6791456 0.83 CCNA2 (0.62) CCNA2CDK2CCNA1IKBKBAURKA
SCHEMBL6794909 0.83 CCNA2 (0.62) CCNA2CDK2CCNA1IKBKBAURKA
SCHEMBL5334053 0.81 CCNA2 (0.62) CCNA2CDK2CCNA1IKBKBAURKA
SCHEMBL6665468 0.80 CCNA2 (0.72) CCNA2CDK2CCNA1IKBKBAURKA
SCHEMBL5337003 0.79 IKBKB (0.60) CCNA2CDK2CCNA1IKBKB
SCHEMBL5227494 0.79 CCNA2 (1.00) CCNA2CDK2CCNA1IKBKB
SCHEMBL6659189 0.78 CCNA2 (0.64) CCNA2CDK2CCNA1IKBKBAURKA
SCHEMBL5334241 0.78 IKBKB (0.58) CCNA2CDK2CCNA1IKBKB
SCHEMBL5335359 0.78 CCNA2 (0.58) CCNA2CDK2CCNA1IKBKBAURKA
SCHEMBL6661725 0.77 CCNA2 (0.71) CCNA2CDK2CCNA1IKBKBAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1476431-A1 TRICYCLIC PYRAZOLE DERIVATIVES FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2004-11-17 EP disclosed
WO-2003070706-A1 TRICYCLIC PYRAZOLE DERIVATIVES FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2003-08-28 WO disclosed