SCHEMBL6664359

SCHEMBL6664359

COc1ccc(OCC(O)CNC2CCN(c3ncnc4scc(-c5ccccc5)c34)CC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 20/20 1.00
ADRB3 P13945 20/20 1.00
ADRB1 P08588 17/20 0.89

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6664389 0.94 ADRB3 (1.00) ADRB2ADRB3ADRB1
SCHEMBL6836550 0.94 ADRB2 (0.89) ADRB2ADRB3ADRB1
SCHEMBL4435801 0.93 ADRB3 (1.00) ADRB2ADRB3ADRB1
SCHEMBL4553648 0.93 ADRB3 (1.00) ADRB2ADRB3ADRB1
SCHEMBL4431300 0.93 ADRB3 (1.00) ADRB2ADRB3ADRB1
SCHEMBL4430206 0.92 ADRB3 (1.00) ADRB2ADRB3ADRB1
SCHEMBL6664332 0.92 ADRB2 (1.00) ADRB2ADRB3ADRB1
SCHEMBL6661634 0.92 ADRB3 (0.89) ADRB2ADRB3ADRB1
SCHEMBL6684421 0.92 ADRB3 (0.84) ADRB2ADRB3ADRB1
SCHEMBL6663555 0.90 ADRB3 (0.87) ADRB2ADRB3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040138238-A1 Substituted aminopyrimidine compounds as neurokinin antagonists PREDIX PHARMACEUTICALS HOLDINGS, INC. 2004-07-15 US claimed
WO-2004014850-A2 SUBSTITUTED AMINOPYRIMIDINES AS NEUROKININ ANTAGONISTS PREDIX PHARMACEUTICALS HOLDINGS, INC. (US) 2004-02-19 WO claimed
US-20040138238-A1 Substituted aminopyrimidine compounds as neurokinin antagonists PREDIX PHARMACEUTICALS HOLDINGS, INC. 2004-07-15 US disclosed
WO-2004014850-A2 SUBSTITUTED AMINOPYRIMIDINES AS NEUROKININ ANTAGONISTS PREDIX PHARMACEUTICALS HOLDINGS, INC. (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040138238-A1 Substituted aminopyrimidine compounds as neurokinin antagonists TACR1, GRPR, BDKRB1 ADRB2 192/4885ADRB3 324/4885ADRB1 136/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.