SCHEMBL6667030

SCHEMBL6667030

Oc1cc(-c2ccccc2)nc2cc(F)ccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 5/20 0.54
ABCG2 Q9UNQ0 1/20 0.46
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
TOP1 P11387 2/20 0.44
CYP19A1 P11511 1/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
KDM4E B2RXH2 2/20 0.44
LMNA P02545 2/20 0.44
PDE10A Q9Y233 1/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ACHE P22303 1/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 1/20 0.43
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
HIF1A Q16665 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6663164 0.89 DHODH (0.53) DHODHESR1ESR2TOP1CYP19A1
SCHEMBL3625999 0.89 DHODH (0.62) DHODHABCG2ESR1ESR2TOP1
SCHEMBL4855755 0.85 CYP19A1 (0.60) DHODHABCG2TOP1CYP19A1SMN1; SMN2
SCHEMBL12201040 0.83 ESR1 (0.53) DHODHESR1ESR2SMN1; SMN2KDM4E
SCHEMBL1256551 0.83 ACHE (0.61) DHODHSMN1; SMN2KDM4ELMNAPDE10A
Methane SCHEMBL10433561 0.81 ACHE (0.59) DHODHSMN1; SMN2KDM4ELMNAPDE10A
SCHEMBL20696076 0.81 ACHE (0.59) DHODHSMN1; SMN2KDM4ELMNAPDE10A
SCHEMBL6660719 0.81 TOP1 (0.58) DHODHABCG2ESR1ESR2TOP1
SCHEMBL16639053 0.81 ACHE (0.47) DHODHESR1ESR2SMN1; SMN2KDM4E
SCHEMBL10155099 0.81 KDM4E (0.56) SMN1; SMN2KDM4ELMNAPDE10AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861864-B1 Method of preparation of polyquinolines HITACHI CHEMICAL CO LTD (JP) 2004-08-25 EP disclosed
EP-0861864-A2 Method of preparation of polyquinolines HITACHI CHEMICAL CO., LTD. (JP) 1998-09-02 EP disclosed
US-5786071-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-07-28 US disclosed
US-5723573-A ACETYLENIC END GROUPS HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-03-03 US disclosed
US-5648448-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1997-07-15 US disclosed