SCHEMBL6668153

SCHEMBL6668153

CCN(CC)C(CCC(C)N)c1nc(Cl)nc2cc(Cl)ccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.35
CYP2D6 P10635 3/20 0.34
PRNP P04156 2/20 0.34
CHRM2 P08172 2/20 0.34
CHRM4 P08173 2/20 0.34
CHRM5 P08912 2/20 0.34
ADRA2A P08913 2/20 0.34
CHRM1 P11229 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
CHRM3 P20309 2/20 0.34
MTOR P42345 2/20 0.34
KCNH2 Q12809 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
CYP2C19 P33261 2/20 0.34
APP P05067 1/20 0.34
NQO2 P16083 1/20 0.34
BACE1 P56817 1/20 0.34
CXCR4 P61073 1/20 0.34
PDE3A Q14432 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5917501 0.83 NPC1 (0.44) NPC1RAB9AMEN1KMT2ANPSR1
SCHEMBL6667631 0.81 RXFP1 (0.31) NR4A2CYP2D6PRNPCHRM2CHRM4
SCHEMBL6667816 0.80 FLT3 (0.42)
SCHEMBL16568037 0.76 NR4A2 (0.46) NR4A2CYP2D6PRNPCHRM2CHRM4
SCHEMBL17799171 0.74 USP2 (0.52) CYP2D6PRNPCHRM2CHRM4CHRM5
SCHEMBL30026121 0.70 NR4A2 (0.44) NR4A2CYP2D6PRNPCHRM2CHRM4
SCHEMBL28887030 0.67 CYP1A2 (0.41) NR4A2CYP2D6CYP1A2NPC1KDM4E
SCHEMBL6672856 0.67 FLT3 (0.46)
SCHEMBL6672860 0.67 FLT3 (0.46)
SCHEMBL3973470 0.67 POLB (0.44) NR4A2HSD17B10POLBKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004030672-A1 USE OF 4 AMINO-QUINAZOLINES AS ANTI CANCER AGENTS MERCK PATENT GMBH (DE) 2004-04-15 WO disclosed
EP-1318984-A1 4-AMINO-QUINAZOLINES MERCK PATENT GmbH (DE) 2003-06-18 EP disclosed
WO-2002024667-A1 4-AMINO-QUINAZOLINES MERCK PATENT GMBH (DE) 2002-03-28 WO disclosed