SCHEMBL6668299

SCHEMBL6668299

CCN(CC)CCCC(C)Nc1nc(-c2cccc(-c3cccnc3)c2)nc2cc(Cl)ccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 3/20 0.56
CSK P41240 1/20 0.53
BTK Q06187 1/20 0.53
ERBB4 Q15303 1/20 0.53
CAMK1G Q96NX5 1/20 0.53
CYP2D6 P10635 3/20 0.52
CHRM2 P08172 3/20 0.52
CHRM4 P08173 3/20 0.52
CHRM5 P08912 3/20 0.52
ADRA2A P08913 3/20 0.52
CHRM1 P11229 3/20 0.52
ADRA2B P18089 3/20 0.52
ADRA2C P18825 3/20 0.52
CHRM3 P20309 3/20 0.52
KCNH2 Q12809 3/20 0.52
PRNP P04156 2/20 0.52
MTOR P42345 2/20 0.52
TDP1 Q9NUW8 2/20 0.52
CYP2C19 P33261 2/20 0.52
TMEM97 Q5BJF2 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6673288 0.86 CCR4 (0.68) CCR4CSKBTKERBB4CAMK1G
SCHEMBL3971151 0.85 CCR4 (0.68) CCR4CSKBTKERBB4CAMK1G
SCHEMBL3975275 0.84 CCR4 (0.63) CCR4CSKBTKERBB4CAMK1G
SCHEMBL3979569 0.82 CCR4 (0.55) CCR4CSKBTKERBB4CAMK1G
SCHEMBL17829849 0.81 CCR4 (0.67) CCR4CSKBTKERBB4CAMK1G
SCHEMBL4269216 0.79 CYP2D6 (0.63) CCR4CSKBTKERBB4CAMK1G
SCHEMBL3975241 0.78 CCR4 (0.51) CCR4CSKBTKERBB4CAMK1G
SCHEMBL17831886 0.78 CCR4 (0.63) CCR4POLBFLT3
SCHEMBL17833178 0.77 CCR4 (0.55) CCR4CSKBTKERBB4CAMK1G
SCHEMBL27599065 0.77 CCR4 (0.56) CCR4CSKBTKERBB4CAMK1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004030672-A1 USE OF 4 AMINO-QUINAZOLINES AS ANTI CANCER AGENTS MERCK PATENT GMBH (DE) 2004-04-15 WO disclosed
EP-1318984-A1 4-AMINO-QUINAZOLINES MERCK PATENT GmbH (DE) 2003-06-18 EP disclosed
WO-2002024667-A1 4-AMINO-QUINAZOLINES MERCK PATENT GMBH (DE) 2002-03-28 WO disclosed