SCHEMBL6668428

SCHEMBL6668428

CCOC(=O)c1c[nH]c(-c2ccc(-c3ccc(N4CC(NC(=O)CC)OC4=O)cc3F)cn2)n1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOA P21397 14/20 0.44
MAOB P27338 2/20 0.44
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
CALML3 P27482 3/20 0.40
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6673572 0.84 MAOA (0.49) MAOAMAOBCYP3A4CYP2C19CALML3
SCHEMBL6646892 0.82 MAOA (0.49) MAOAMAOBCYP3A4CYP2C19CALML3
SCHEMBL6646472 0.81 MAOA (0.51) MAOAMAOBCYP3A4CYP2C19CALML3
SCHEMBL6644071 0.80 MAOA (0.52) MAOAMAOBCYP3A4CYP2C19CALML3
SCHEMBL6643168 0.80 CALML3 (0.49) MAOAMAOBCYP3A4CYP2C19CALML3
SCHEMBL6642847 0.79 MAOA (0.53) MAOAMAOBCYP3A4CYP2C19CALML3
SCHEMBL6641386 0.78 MAOA (0.52) MAOAMAOBCYP3A4CYP2C19CALML3
SCHEMBL6646270 0.78 MAOA (0.47) MAOAMAOBCYP3A4CYP2C19CALML3
SCHEMBL6644478 0.78 CALML3 (0.47) MAOAMAOBCYP3A4CYP2C19CALML3
SCHEMBL6668137 0.77 CALML3 (0.42) MAOAMAOBCYP3A4CYP2C19CALML3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289984-A4 NOVEL OXAZOLIDINONE DERIVATIVES AND A PROCESS FOR THE PREPARATION THEREOF DONG A PHARM CO LTD (KR) 2004-11-24 EP disclosed
EP-1289984-A1 NOVEL OXAZOLIDINONE DERIVATIVES AND A PROCESS FOR THE PREPARATION THEREOF Dong A Pharmaceutical Co. Ltd. (KR) 2003-03-12 EP disclosed
WO-2001094342-A1 NOVEL OXAZOLIDINONE DERIVATIVES AND A PROCESS FOR THE PREPARATION THEREOF DONG A PHARM. CO., LTD. (KR) 2001-12-13 WO disclosed