SCHEMBL6671672

SCHEMBL6671672

CCc1nn(C)c(CC)c1Oc1c(C#N)cccc1C#N

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RARG P13631 1/20 0.41
RORC P51449 1/20 0.41
MAPT P10636 2/20 0.33
CYP11B2 P19099 1/20 0.33
GAA P10253 1/20 0.33
PDE10A Q9Y233 1/20 0.31
GRIA2 P42262 1/20 0.31
GRIA4 P48058 1/20 0.31
PGR P06401 4/20 0.31
NPSR1 Q6W5P4 1/20 0.31
GCK P35557 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL509344 0.79 KCNH2 (0.41) RARGRORCCYP11B2GRIA2GRIA4
SCHEMBL4105490 0.78 PGR (0.52) RARGRORCCYP11B2PGR
SCHEMBL10254059 0.68 KCNH2 (0.44) RARGRORCCYP11B2PGR
SCHEMBL4112493 0.65 PGR (0.42) PGR
SCHEMBL4106530 0.64 PGR (0.49) CYP11B2PGR
SCHEMBL4115324 0.64 PGR (0.49) CYP11B2PGR
SCHEMBL2752305 0.64 MAPT (0.33) MAPTGAANPSR1
SCHEMBL2752424 0.64 KDM4E (0.34) MAPTGAANPSR1GCK
SCHEMBL15687305 0.63 PDE5A (0.37) MAPT
SCHEMBL15388910 0.63 TSHR (0.41) MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377556-A1 PYRAZOLE DERIVATIVES FOR TREATING HIV Pfizer Limited (GB) 2004-01-07 EP disclosed
WO-2002085860-A1 PYRAZOLE DERIVATIVES FOR TREATING HIV PFIZER LIMITED (GB) 2002-10-31 WO disclosed