SCHEMBL6671694

SCHEMBL6671694

COC(=O)CC(NC(=O)CNC(=O)CCCNc1cc(C)ccn1)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 8/20 0.54
ITGB6 P18564 8/20 0.54
ITGB3 P05106 7/20 0.54
ITGB5 P18084 7/20 0.54
ITGA2B P08514 4/20 0.52
ITGB1 P05556 1/20 0.49
ITGA5 P08648 1/20 0.49
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
POLB P06746 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
LMNA P02545 2/20 0.43
ALDH1A1 P00352 3/20 0.42
HPGD P15428 1/20 0.42
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7173698 0.98 ITGAV (0.54) ITGAVITGB6ITGB3ITGB5ITGA2B
SCHEMBL7171933 0.93 ITGAV (0.54) ITGAVITGB6ITGB3ITGB5ITGA2B
SCHEMBL6669951 0.92 ITGAV (0.61) ITGAVITGB6ITGB3ITGB5ITGA2B
SCHEMBL7171785 0.90 ITGAV (0.55) ITGAVITGB6ITGB3ITGB5ITGA2B
SCHEMBL7177374 0.90 ITGAV (0.52) ITGAVITGB6ITGB3ITGB5ITGA2B
SCHEMBL7172069 0.90 ITGAV (0.64) ITGAVITGB6ITGB3ITGB5ITGA2B
SCHEMBL7172197 0.89 ITGAV (0.63) ITGAVITGB6ITGB3ITGB5ITGA2B
SCHEMBL7172208 0.89 ITGAV (0.63) ITGAVITGB6ITGB3ITGB5ITGA2B
SCHEMBL7172201 0.89 ITGAV (0.54) ITGAVITGB6ITGB3ITGB5ITGA2B
SCHEMBL7172214 0.89 ITGAV (0.63) ITGAVITGB6ITGB3ITGB5ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153014-B1 BETA-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2004-09-22 EP disclosed
US-6576637-B1 Such as 3-(4-methyl-3-nitrophenyl)-3-(2-(4-(pyridin-2-yl-amino)butyryl amino)acetylamino)propionic acid; thrombosis, heart infarct, coronary heart diseases, arteriosclerosis, inflammations, MERCK PATENT GMBH (DE) 2003-06-10 US disclosed