SCHEMBL7177374

SCHEMBL7177374

COC(=O)CC(NC(=O)CNC(=O)CCCNc1ccccn1)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 17/20 0.52
ITGB3 P05106 16/20 0.52
ITGB6 P18564 5/20 0.52
ITGB5 P18084 5/20 0.52
ITGA2B P08514 5/20 0.52
LMNA P02545 1/20 0.48
ITGB1 P05556 1/20 0.38
ITGA5 P08648 1/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7176745 0.97 ITGB3 (0.56) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7169953 0.91 ITGAV (0.64) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6671694 0.90 ITGAV (0.54) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7168458 0.90 ITGAV (0.54) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7168475 0.90 ITGAV (0.63) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7168468 0.90 ITGAV (0.63) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7168452 0.90 ITGAV (0.63) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7173599 0.89 ITGAV (0.48) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7171242 0.88 ITGB3 (0.68) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7173698 0.88 ITGAV (0.54) ITGAVITGB3ITGB6ITGB5ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6576637-B1 Such as 3-(4-methyl-3-nitrophenyl)-3-(2-(4-(pyridin-2-yl-amino)butyryl amino)acetylamino)propionic acid; thrombosis, heart infarct, coronary heart diseases, arteriosclerosis, inflammations, MERCK PATENT GMBH (DE) 2003-06-10 US disclosed
EP-1153014-A2 BETA-ALANINE DERIVATIVES MERCK PATENT GmbH (DE) 2001-11-14 EP disclosed
WO-2000048996-A2 β-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2000-08-24 WO disclosed