SCHEMBL6675381

SCHEMBL6675381

CCN=C(N)Nc1cccc(CN)c1OC

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 3/20 0.45
CACNA1C Q13936 2/20 0.45
PTGIR P43119 2/20 0.42
SIGMAR1 Q99720 5/20 0.40
GRIN2D O15399 3/20 0.40
GRIN3B O60391 3/20 0.40
GRIN1 Q05586 3/20 0.40
GRIN2A Q12879 3/20 0.40
GRIN2B Q13224 3/20 0.40
GRIN2C Q14957 3/20 0.40
GRIN3A Q8TCU5 3/20 0.40
CXCR4 P61073 2/20 0.33
NOS1 P29475 2/20 0.33
GLS O94925 1/20 0.33
NOS3 P29474 1/20 0.33
NOS2 P35228 1/20 0.33
CASR P41180 1/20 0.33
HTR7 P34969 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6680717 0.99 SCN5A (0.44) SCN5ACACNA1CPTGIRSIGMAR1GRIN2D
SCHEMBL6675317 0.82 CACNA1C (0.49) SCN5ACACNA1CPTGIRSIGMAR1GRIN2D
Hydrochloric Acid SCHEMBL6674250 0.81 CACNA1C (0.48) SCN5ACACNA1CPTGIRSIGMAR1GRIN2D
SCHEMBL6676349 0.81 CACNA1C (0.48) SCN5ACACNA1CPTGIRSIGMAR1GRIN2D
SCHEMBL6676424 0.81 CACNA1C (0.48) SCN5ACACNA1CPTGIRSIGMAR1GRIN2D
Hydrochloric Acid SCHEMBL6675369 0.80 CACNA1C (0.47) SCN5ACACNA1CPTGIRSIGMAR1GRIN2D
SCHEMBL6678288 0.78 PTGIR (0.40) SCN5ACACNA1CPTGIRSIGMAR1GRIN2D
SCHEMBL6676191 0.78 CACNA1C (0.45) SCN5ACACNA1CPTGIRSIGMAR1GRIN2D
Hydrochloric Acid SCHEMBL6679059 0.77 CACNA1C (0.44) SCN5ACACNA1CPTGIRSIGMAR1GRIN2D
SCHEMBL6676762 0.75 GLS (0.35) SCN5ACACNA1CGLSCASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP claimed