SCHEMBL6676211

SCHEMBL6676211

COc1ccc(NC(N)=S)cc1C(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
GAA P10253 2/20 0.58
IMPDH2 P12268 1/20 0.46
IMPDH1 P20839 1/20 0.46
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDM4E B2RXH2 2/20 0.42
P2RX5 Q93086 1/20 0.41
P2RX4 Q99571 1/20 0.41
P2RX7 Q99572 1/20 0.41
P2RX2 Q9UBL9 1/20 0.41
KMT2A Q03164 4/20 0.40
MAPT P10636 3/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
CXCR2 P25025 2/20 0.38
MEN1 O00255 2/20 0.38
RAB9A P51151 2/20 0.38
CA12 O43570 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678137 0.82 C5AR1 (0.46) ALDH1A1GAACYP2C9KDM4EP2RX4
SCHEMBL6686878 0.79 KDM4E (0.44) ALDH1A1GAAIMPDH2IMPDH1KDM4E
SCHEMBL7247258 0.79 ALDH1A1 (0.56) ALDH1A1GAAIMPDH2IMPDH1CYP1A2
SCHEMBL6679990 0.78 ALDH1A1 (0.55) ALDH1A1GAAIMPDH2IMPDH1CYP1A2
SCHEMBL6678276 0.78 ALDH1A1 (0.49) ALDH1A1GAACYP1A2KMT2ASMN1; SMN2
SCHEMBL6679066 0.77 ALDH1A1 (0.54) ALDH1A1GAAKMT2A
SCHEMBL10809983 0.76 ALDH1A1 (0.72) ALDH1A1GAAIMPDH2IMPDH1CYP1A2
SCHEMBL14499383 0.76 GAA (0.54) ALDH1A1GAAIMPDH2IMPDH1CYP1A2
SCHEMBL12071196 0.75 CYP17A1 (0.51) ALDH1A1GAACYP2C9CYP2C19KMT2A
SCHEMBL6676215 0.75 KDM4E (0.41) ALDH1A1GAAIMPDH2IMPDH1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed