SCHEMBL6676219

SCHEMBL6676219

O=c1[nH]cc(-c2ccccn2)c(-c2ccccn2)c1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.43
L3MBTL1 Q9Y468 5/20 0.43
ALDH1A1 P00352 4/20 0.43
TDP1 Q9NUW8 4/20 0.43
HSP90AA1 P07900 2/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CHEK1 O14757 1/20 0.42
LMNA P02545 6/20 0.41
KDM4E B2RXH2 6/20 0.41
HIF1A Q16665 2/20 0.41
POLB P06746 2/20 0.41
CCR1 P32246 2/20 0.41
CCR5 P51681 2/20 0.41
CCR8 P51685 2/20 0.41
CYP1A2 P05177 1/20 0.41
METAP1 P53582 1/20 0.41
BLM P54132 1/20 0.41
DOHH Q9BU89 1/20 0.41
P4HTM Q9NXG6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18074831 0.91 PARP1 (0.41) HTTL3MBTL1ALDH1A1TDP1HSP90AA1
SCHEMBL6679170 0.85 CYP2A6 (0.54) HTTL3MBTL1ALDH1A1TDP1HSP90AA1
SCHEMBL3667468 0.79 PARP1 (0.45) HTTL3MBTL1ALDH1A1CHEK1LMNA
SCHEMBL8675092 0.73 ALDH1A1 (0.56) HTTL3MBTL1ALDH1A1TDP1CHEK1
SCHEMBL787084 0.73 PRKCI (0.51) HTTL3MBTL1ALDH1A1TDP1HSP90AA1
SCHEMBL6679876 0.72 PADI4 (0.41) HTTL3MBTL1ALDH1A1KMT2ACHEK1
SCHEMBL2763150 0.72 CDC7 (0.39) HTTL3MBTL1ALDH1A1KMT2ANPSR1
SCHEMBL3667347 0.72 MAPK14 (0.42) HTTALDH1A1CHEK1KDM4EMAPT
SCHEMBL6674838 0.72 CYP2A6 (0.55) P4HTMNPC1RAB9ASMN1; SMN2HPGD
SCHEMBL1888457 0.71 PRMT5 (0.43) HTTL3MBTL1ALDH1A1TDP1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465626-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES Eisai Co., Ltd. (JP) 2004-10-13 EP disclosed
WO-2003047577-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES EISAI CO LTD (JP) 2003-06-12 WO disclosed