SCHEMBL6676802

SCHEMBL6676802

CC(C)(C)OC(=O)NN(Cc1cccc(N)c1)C(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.55
CTSL P07711 2/20 0.42
CTSB P07858 2/20 0.42
CTSS P25774 2/20 0.42
PTGES O14684 1/20 0.40
HSD11B1 P28845 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
GLS O94925 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA7 P43166 1/20 0.37
CA14 Q9ULX7 1/20 0.37
KCNQ4 P56696 1/20 0.35
KCNQ5 Q9NR82 1/20 0.35
BACE1 P56817 3/20 0.35
SLC7A5 Q01650 1/20 0.35
NQO2 P16083 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1402743 0.84 AKT1 (0.57) AKT1CTSLCTSBCTSSSLC7A5
SCHEMBL2394937 0.83 AKT1 (0.53) AKT1CTSLCTSBCTSSSLC7A5
SCHEMBL6681292 0.82 AKT1 (0.49) AKT1CTSLCTSBCTSSPTGES
SCHEMBL7247305 0.81 GRM2 (0.43) AKT1HSD11B1HDAC3HDAC1HDAC2
SCHEMBL6681909 0.81 AKT1 (0.51) AKT1
SCHEMBL6675521 0.81 HDAC3 (0.53) AKT1CTSLCTSBCTSSPTGES
SCHEMBL2228851 0.80 HSD11B1 (0.51) CTSLCTSBCTSSHSD11B1GLS
SCHEMBL1403248 0.80 AKT1 (0.53) AKT1CTSLCTSBCTSSSLC7A5
SCHEMBL396085 0.79 HSD11B1 (0.41) AKT1HSD11B1HDAC3HDAC1HDAC2
SCHEMBL6681914 0.78 HDAC1 (0.45) PTGESHSD11B1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed