SCHEMBL6677086

SCHEMBL6677086

CCOC(=O)c1cc(S(=O)(=O)c2ccc(CCNC(C(=O)OC(C)(C)C)[C@H](O)c3cccc(Cl)c3)cc2)ccc1[N+](=O)[O-]

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.36
LMNA P02545 4/20 0.36
NPSR1 Q6W5P4 3/20 0.36
HTT P42858 3/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
ADRB3 P13945 5/20 0.35
ADRB1 P08588 2/20 0.35
ADRB2 P07550 1/20 0.35
THRB P10828 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GPR55 Q9Y2T6 1/20 0.34
CA2 P00918 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6680679 0.89 ADRB3 (0.36) HTTADRB3ADRB1ADRB2CA2
SCHEMBL6677699 0.88 ADRB3 (0.37) LMNAADRB3ADRB1ADRB2CA2
SCHEMBL6677357 0.87 ADRB3 (0.37) LMNAADRB3ADRB1ADRB2CA2
SCHEMBL6681115 0.87 ADRB3 (0.37) MAPTLMNAKMT2AMEN1ADRB3
SCHEMBL6677162 0.85 ADRB3 (0.35) MAPTLMNANPSR1KMT2AMEN1
SCHEMBL6676709 0.85 MEN1 (0.32) MAPTLMNANPSR1HTTKMT2A
SCHEMBL6680598 0.82 ADRB3 (0.40) ADRB3ADRB1ADRB2CA2
SCHEMBL6679366 0.82 ADRB3 (0.39) ADRB3ADRB1ADRB2CA2
SCHEMBL6680863 0.82 ADRB3 (0.47) MAPTLMNAKMT2AMEN1ADRB3
SCHEMBL6676373 0.81 ADRB3 (0.40) ADRB3ADRB1ADRB2CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004045610-A1 AMINOALCOHOL DERIVATIVES AND THEIR USE AS BETA-3 ADRENERGIC RECEPTOR AGONISTS FUJISAWA PHARMACEUTICAL CO., LTD (JP) 2004-06-03 WO disclosed