SCHEMBL6678239

SCHEMBL6678239

Cc1ccc(N2C(=O)c3ccccc3C2=O)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
ADCY2 Q08462 1/20 0.51
GRM1 Q13255 4/20 0.50
GRM4 Q14833 2/20 0.50
NR1H3 Q13133 2/20 0.48
SCN2A Q99250 1/20 0.45
CYP3A4 P08684 1/20 0.45
NFKB1 P19838 1/20 0.45
PMP22 Q01453 1/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
GRM8 O00222 1/20 0.44
GRM5 P41594 1/20 0.44
GRM7 Q14831 1/20 0.44
PGR P06401 1/20 0.44
NR1H2 P55055 1/20 0.44
ELANE P08246 1/20 0.43
GAA P10253 1/20 0.43
TLR9 Q9NR96 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30273450 1.00 ESR1 (0.53) ESR1ESR2ADCY2GRM1GRM4
SCHEMBL10626656 0.82 ESR1 (0.56) ESR1ESR2GRM1GRM4SCN2A
SCHEMBL28665183 0.82 ESR1 (0.56) ESR1ESR2GRM1GRM4NR1H3
SCHEMBL14339993 0.79 CA1 (0.47) ESR1ESR2ADCY2GRM1GRM4
SCHEMBL7729256 0.79 MEN1 (0.53) ESR1ESR2GRM1GRM4SCN2A
SCHEMBL30273429 0.79 MEN1 (0.53) ESR1ESR2GRM1GRM4SCN2A
SCHEMBL5924351 0.79 CYP3A4 (0.66) ESR1ESR2GRM1GRM4NR1H3
SCHEMBL15199351 0.79 CA1 (0.43) ESR1ESR2ADCY2GRM1GRM4
SCHEMBL7514060 0.79 MEN1 (0.49) ESR1ESR2NR1H3SCN2ACYP3A4
SCHEMBL3106326 0.79 SCN2A (0.68) ESR1ESR2GRM1GRM4NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115701423-A Preparation method of trifluoroethyl sulfide (sulfoxide) substituted benzene compound and intermediate thereof 沈阳化工大学 2023-02-10 CN disclosed
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed