SCHEMBL6678259

SCHEMBL6678259

CC(C)(C)OC(=O)NC(C)(C)c1cccc(NC(N)=S)c1OCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.40
HDAC1 Q13547 1/20 0.39
LMNA P02545 2/20 0.39
POLB P06746 1/20 0.39
LTA4H P09960 1/20 0.37
CTSS P25774 1/20 0.37
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
SYK P43405 1/20 0.36
CYP2C9 P11712 1/20 0.36
PTGER1 P34995 1/20 0.36
PPARA Q07869 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28747641 0.83 HDAC1 (0.40) BRD4HDAC1LMNAPOLBLTA4H
SCHEMBL6675988 0.83 HDAC1 (0.43) HDAC1LMNALTA4HCTSSMEN1
SCHEMBL6680185 0.82 BCHE (0.38) BRD4HDAC1LMNAPOLBLTA4H
SCHEMBL27478367 0.81 GAA (0.41) BRD4LMNAPOLBMEN1GAA
SCHEMBL6680187 0.80 BRD4 (0.39) BRD4HDAC1LMNAPOLBCTSS
SCHEMBL6678137 0.80 C5AR1 (0.46) LMNALTA4HMEN1GAAKMT2A
SCHEMBL6677550 0.78 HTR1A (0.47) POLBMEN1KMT2ASMN1; SMN2
SCHEMBL30705048 0.77 BRD4 (0.54) BRD4HDAC1MEN1KMT2ASYK
SCHEMBL6680190 0.74 SYK (0.35) LTA4HCTSSMEN1KMT2ASYK
SCHEMBL28870996 0.73 BRD4 (0.52) BRD4MEN1KMT2ACYP2C9PTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed