SCHEMBL6679321

SCHEMBL6679321

COc1cc(C)ccc1N1C(=O)c2ccccc2C1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.54
SCN2A Q99250 1/20 0.54
NR1H3 Q13133 4/20 0.52
ESR1 P03372 1/20 0.52
GRM1 Q13255 1/20 0.52
GRM4 Q14833 1/20 0.52
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
NR1H2 P55055 2/20 0.49
CASP6 P55212 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HTT P42858 1/20 0.49
ADCY2 Q08462 1/20 0.48
GAA P10253 2/20 0.48
CASP3 P42574 1/20 0.48
SENP8 Q96LD8 1/20 0.48
SENP7 Q9BQF6 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6968611 0.84 G6PD (0.59) KMT2AMEN1SCN2ANR1H3ESR1
SCHEMBL11808285 0.84 ESR1 (0.72) KMT2AMEN1SCN2ANR1H3ESR1
SCHEMBL10915309 0.83 CYP3A4 (0.60) KMT2AMEN1SCN2ANR1H3ESR1
SCHEMBL30758650 0.81 KMT2A (0.76) KMT2AMEN1SCN2ANR1H3NR1H2
SCHEMBL29168849 0.81 KMT2A (0.76) KMT2AMEN1SCN2ANR1H3NR1H2
SCHEMBL28665183 0.80 ESR1 (0.56) KMT2AMEN1NR1H3ESR1GRM1
SCHEMBL6676243 0.79 NR1H3 (0.57) KMT2AMEN1SCN2ANR1H3ESR1
SCHEMBL7451753 0.79 NPC1 (0.49) SCN2ANR1H3NPC1RAB9ASMN1; SMN2
SCHEMBL16592564 0.78 RECQL (0.62) KMT2AMEN1SCN2ANR1H3ESR1
SCHEMBL30758606 0.78 RECQL (0.62) KMT2AMEN1SCN2ANR1H3ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed