SCHEMBL6680592

SCHEMBL6680592

COC(=O)Cc1ccc(CN(c2ccc(Cl)c(Cl)c2)c2nnc(-c3cccc(Oc4cccc(C(F)(F)F)c4)c3)s2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
HPGD P15428 3/20 0.40
HSD17B10 Q99714 3/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CACNA1B Q00975 1/20 0.38
S1PR1 P21453 3/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
P2RY1 P47900 1/20 0.36
MEN1 O00255 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KDM4E B2RXH2 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PPARA Q07869 2/20 0.36
PPARG P37231 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6154582 0.92 CETP (0.41) LMNAHPGDHSD17B10NPC1MAPT
SCHEMBL6155264 0.90 CETP (0.40) LMNAHPGDHSD17B10NPC1MAPT
SCHEMBL6153971 0.89 S1PR1 (0.40) LMNAHPGDHSD17B10NPC1CACNA1B
SCHEMBL6155267 0.88 HSD17B10 (0.40) LMNAHPGDHSD17B10NPC1CACNA1B
SCHEMBL6154990 0.87 P2RY1 (0.40) LMNAHPGDHSD17B10NPC1MAPT
SCHEMBL6155070 0.80 PTPN5 (0.45) LMNAHPGDHSD17B10NPC1ROCK2
SCHEMBL6155036 0.80 HSD17B10 (0.38) LMNAHPGDHSD17B10NPC1S1PR1
SCHEMBL6154034 0.79 KMO (0.47) LMNAHPGDHSD17B10NPC1ROCK2
SCHEMBL6154252 0.78 GCGR (0.39) LMNAHPGDHSD17B10NPC1MAPT
SCHEMBL4955510 0.77 NR1H2 (0.38) LMNAHPGDHSD17B10NPC1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1446110-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES Structural Bioinformatics Inc. (US) 2004-08-18 EP disclosed
WO-2003032916-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES STRUCTURAL BIOINFORMATICS INC. (US) 2003-04-24 WO disclosed