SCHEMBL6680801

SCHEMBL6680801

CCOC(=O)c1cccc(Oc2ccc(S(=O)(=O)c3ccc(CCCNC(Cc4ccccc4)[C@H](O)c4cccc(Cl)c4)cc3)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 13/20 0.46
ADRB1 P08588 9/20 0.42
CYP4F2 P78329 1/20 0.39
CYP4A11 Q02928 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 2/20 0.39
SLC2A1 P11166 1/20 0.38
LPAR1 Q92633 1/20 0.38
LPAR5 Q9H1C0 1/20 0.38
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6681933 0.96 ADRB3 (0.42) ADRB3ADRB1CYP4F2CYP4A11MEN1
SCHEMBL6677081 0.92 CYP4F2 (0.42) ADRB3ADRB1CYP4F2CYP4A11MEN1
SCHEMBL6677033 0.90 ADRB3 (0.44) ADRB3ADRB1CYP4F2CYP4A11ALDH1A1
Hydrochloric Acid SCHEMBL6803942 0.86 ADRB3 (0.43) ADRB3ADRB1CYP4F2CYP4A11MEN1
SCHEMBL6687818 0.85 ADRB3 (0.39) ADRB3ADRB1MEN1KMT2AMAPT
SCHEMBL6679530 0.85 ADORA1 (0.38) ADRB3ADRB1KMT2AMAPTSLC2A1
Hydrochloric Acid SCHEMBL6679835 0.83 ADRB3 (0.62) ADRB3ADRB1
Hydrochloric Acid SCHEMBL6679838 0.83 ADRB3 (0.62) ADRB3ADRB1
SCHEMBL6676287 0.83 ADRB3 (0.55) ADRB3ADRB1LPAR1LPAR5
SCHEMBL6676594 0.83 ADRB3 (0.42) ADRB3ADRB1SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004045610-A1 AMINOALCOHOL DERIVATIVES AND THEIR USE AS BETA-3 ADRENERGIC RECEPTOR AGONISTS FUJISAWA PHARMACEUTICAL CO., LTD (JP) 2004-06-03 WO disclosed