SCHEMBL6681035

SCHEMBL6681035

CC/N=C(/NC(=O)OC(C)(C)C)Nc1ccc(OCc2ccccc2)c(C(C)(C)NC(=O)OC(C)(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 9/20 0.40
BCHE P06276 1/20 0.39
CNR2 P34972 1/20 0.39
CYP2C9 P11712 1/20 0.39
PTGER1 P34995 1/20 0.39
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
MAPKAPK2 P49137 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LTA4H P09960 1/20 0.36
CYP19A1 P11511 1/20 0.36
ACP1 P24666 1/20 0.36
PTPN12 Q05209 1/20 0.36
PTPN13 Q12923 1/20 0.36
SSU72 Q9NP77 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6680473 0.84 CYP2C9 (0.42) C5AR1BCHECNR2CYP2C9PTGER1
SCHEMBL6681039 0.84 C5AR1 (0.39) C5AR1BCHECNR2CYP2C9PTGER1
SCHEMBL27547572 0.82 CYP2C9 (0.42) C5AR1CYP2C9PTGER1MEN1KMT2A
SCHEMBL6678137 0.82 C5AR1 (0.46) C5AR1CYP2C9PTGER1MEN1KMT2A
SCHEMBL6680185 0.81 BCHE (0.38) BCHECNR2CYP2C9PTGER1MEN1
SCHEMBL27544860 0.80 PTGER1 (0.42) C5AR1CYP2C9PTGER1MEN1KMT2A
SCHEMBL6678655 0.78 C5AR1 (0.48) C5AR1MEN1KMT2A
SCHEMBL6680546 0.77 RXFP1 (0.42) MEN1KMT2ASMN1; SMN2
SCHEMBL6678649 0.77 CTSV (0.41) C5AR1CYP2C9PTGER1MEN1KMT2A
SCHEMBL6675702 0.77 CYP2C9 (0.43) BCHECNR2CYP2C9PTGER1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed