SCHEMBL6681763

SCHEMBL6681763

N[C@](CCCNC1CCCc2cccnc21)(C(=O)O)C(=O)c1ccc(CNCc2ccccn2)nc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
CXCR4 P61073 12/20 0.40
CYP3A4 P08684 3/20 0.38
CYP2D6 P10635 3/20 0.38
SLC40A1 Q9NP59 1/20 0.35
HPGD P15428 2/20 0.35
RECQL P46063 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ROCK2 O75116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6691016 0.91 HDAC1 (0.39) HDAC1HDAC6CXCR4CYP3A4CYP2D6
SCHEMBL6018435 0.81 HDAC1 (0.47) HDAC1HDAC6CXCR4CYP3A4CYP2D6
SCHEMBL6018210 0.74 CXCR4 (0.39) HDAC1HDAC6CXCR4SLC40A1
SCHEMBL6019179 0.74 HDAC1 (0.55) HDAC1HDAC6CXCR4CYP3A4CYP2D6
SCHEMBL7024499 0.74 HDAC1 (0.42) HDAC1HDAC6CXCR4CYP3A4CYP2D6
SCHEMBL6687600 0.72 HDAC1 (0.41) HDAC1HDAC6CXCR4CYP3A4CYP2D6
SCHEMBL1874122 0.72 HDAC1 (0.63) HDAC1HDAC6CXCR4CYP3A4CYP2D6
SCHEMBL29823204 0.72 HDAC1 (0.63) HDAC1HDAC6CXCR4CYP3A4CYP2D6
SCHEMBL4065365 0.72 HDAC1 (0.74) HDAC1HDAC6CXCR4HPGDMEN1
SCHEMBL1882612 0.72 HDAC1 (0.62) HDAC1HDAC6CXCR4CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound KUREHA CORPORATION (JP) 2004-08-12 US disclosed
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound CXCR4, CXCR1, CXCR2 HDAC1 1092/4885HDAC6 1799/4885CXCR4 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.