SCHEMBL6682903

SCHEMBL6682903

COc1ccc(-n2nc(C(F)(F)F)nc2-c2ccc(OCCCO)cc2)cn1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 6/20 0.47
PTGS2 P35354 6/20 0.47
MCHR1 Q99705 1/20 0.36
OXTR P30559 3/20 0.36
AVPR2 P30518 2/20 0.36
AVPR1A P37288 2/20 0.36
MALT1 Q9UDY8 2/20 0.35
ABL1 P00519 1/20 0.35
DYRK3 O43781 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
DYRK1A Q13627 1/20 0.34
DYRK2 Q92630 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
MGAT2 Q10469 1/20 0.34
AGER Q15109 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6684307 0.89 PTGS2 (0.47) PTGS1PTGS2OXTRAVPR2AVPR1A
SCHEMBL6681239 0.88 PTGS1 (0.64) PTGS1PTGS2MCHR1OXTRAVPR2
SCHEMBL6682106 0.88 PTGS2 (0.60) PTGS1PTGS2MALT1
SCHEMBL6132606 0.87 PTGS2 (0.57) PTGS1PTGS2OXTRAVPR2AVPR1A
SCHEMBL6687455 0.86 PTGS2 (0.42) PTGS1PTGS2MALT1
SCHEMBL6686275 0.85 PTGS2 (0.43) PTGS1PTGS2MALT1DYRK3CDK2
SCHEMBL6680327 0.84 PTGS1 (0.45) PTGS1PTGS2OXTRAVPR2AVPR1A
SCHEMBL6689709 0.83 PTGS1 (0.46) PTGS1PTGS2OXTRAVPR2AVPR1A
SCHEMBL6132382 0.80 PTGS2 (0.57) PTGS1PTGS2
SCHEMBL6689504 0.79 PTGS1 (0.49) PTGS1PTGS2OXTRAVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060367-A1 IMIDAZOLE AND TRIAZOLE DERIVATIVES USEFUL AS SELECTIVE COX-1 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-07-22 WO disclosed