SCHEMBL6683341

SCHEMBL6683341

COc1ccc(-n2nc(C(F)(F)F)nc2-c2ccc(OCc3ccccc3)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 5/20 0.58
PTGS2 P35354 5/20 0.58
L3MBTL1 Q9Y468 3/20 0.47
GABRA1 P14867 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
GABRA2 P47869 1/20 0.46
ADORA3 P0DMS8 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
MDM2 Q00987 2/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6689709 0.89 PTGS1 (0.46) PTGS1PTGS2L3MBTL1GABRA1GABRG2
SCHEMBL5865649 0.87 PTGS2 (0.60) PTGS1PTGS2L3MBTL1NPC1RAB9A
SCHEMBL6132473 0.86 PTGS2 (0.67) PTGS1PTGS2L3MBTL1SMN1; SMN2MAPT
SCHEMBL6681657 0.84 PTGS1 (0.52) PTGS1PTGS2L3MBTL1GABRA1GABRG2
SCHEMBL6681240 0.82 PTGS2 (0.60) PTGS1PTGS2L3MBTL1HIF1ANPSR1
SCHEMBL6132192 0.82 PTGS2 (0.63) PTGS1PTGS2L3MBTL1HPGDHIF1A
SCHEMBL6132484 0.82 PTGS2 (0.63) PTGS1PTGS2L3MBTL1HPGDHIF1A
SCHEMBL6684663 0.82 PTGS1 (0.62) PTGS1PTGS2L3MBTL1GABRA1GABRG2
SCHEMBL28806023 0.81 PTGS2 (0.60) PTGS1PTGS2L3MBTL1HIF1ANPSR1
SCHEMBL27905338 0.81 PTGS2 (0.60) PTGS1PTGS2L3MBTL1HIF1ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060367-A1 IMIDAZOLE AND TRIAZOLE DERIVATIVES USEFUL AS SELECTIVE COX-1 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-07-22 WO disclosed