SCHEMBL6684012

SCHEMBL6684012

CC(C)(C)OC(=O)ON(Cc1ccc(/C(N)=N\OCc2ccc(F)cc2)cc1)OC(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.37
RAB9A P51151 2/20 0.37
PKM P14618 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
S1PR1 P21453 2/20 0.37
MAOB P27338 2/20 0.35
PARP10 Q53GL7 1/20 0.35
KCNQ4 P56696 1/20 0.34
KCNQ5 Q9NR82 1/20 0.34
NR4A2 P43354 1/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
KMT2A Q03164 1/20 0.32
RIPK1 Q13546 2/20 0.32
GRM2 Q14416 1/20 0.32
NR1D1 P20393 1/20 0.32
CA12 O43570 1/20 0.32
HDAC3 O15379 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7062273 0.96 SMN1; SMN2 (0.39) NPC1RAB9APKMSMN1; SMN2S1PR1
SCHEMBL7062282 0.96 SMN1; SMN2 (0.39) NPC1RAB9APKMSMN1; SMN2S1PR1
SCHEMBL6650316 0.74 SMN1; SMN2 (0.44) NPC1RAB9APKMSMN1; SMN2S1PR1
Isobutane SCHEMBL7062276 0.71 NPC1 (0.46) NPC1RAB9APKMSMN1; SMN2S1PR1
SCHEMBL18740536 0.70 RIPK1 (0.44) KCNQ4KCNQ5CTSSCTSKRIPK1
Ammonia Solution, Strong SCHEMBL6905116 0.69 SMN1; SMN2 (0.39) NPC1RAB9APKMSMN1; SMN2S1PR1
Hydrochloric Acid SCHEMBL6794609 0.68 MAOB (0.51) NPC1RAB9APKMSMN1; SMN2S1PR1
Hydrochloric Acid SCHEMBL6672174 0.68 MAOB (0.51) NPC1RAB9APKMSMN1; SMN2S1PR1
SCHEMBL8363482 0.66 HDAC3 (0.40) NPC1RAB9ASMN1; SMN2GRM2HDAC3
SCHEMBL18763349 0.66 RIPK1 (0.43) KCNQ4KCNQ5CTSSCTSKRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1482940-A2 PRODRUGS OF SUBSTITUTED POLYCYCLIC COMPOUNDS USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE Pharmacia Corporation (US) 2004-12-08 EP disclosed
WO-2003028729-A2 PRODRUGS OF SUBSTITUTED POLYCYCLIC COMPOUNDS USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2003-04-10 WO disclosed