SCHEMBL6684701

SCHEMBL6684701

O=C(O)COCc1cccc(C(F)(F)F)c1-c1cccc(-c2nnc(Nc3ccc(Cl)c(Cl)c3)s2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.42
ROCK1 Q13464 3/20 0.42
GUSB P08236 2/20 0.41
DHODH Q02127 3/20 0.40
BLM P54132 5/20 0.39
S1PR1 P21453 1/20 0.39
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
DNMT1 P26358 1/20 0.36
HTT P42858 1/20 0.36
DUSP3 P51452 1/20 0.36
CACNA1B Q00975 1/20 0.36
APBA1 Q02410 1/20 0.36
MCL1 Q07820 1/20 0.36
WRN Q14191 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6154319 0.75 ROCK1 (0.45) ROCK2ROCK1GUSBDHODHBLM
SCHEMBL6155161 0.71 GUSB (0.60) ROCK2ROCK1GUSBBLMKMT2A
SCHEMBL6153472 0.70 GUSB (0.53) ROCK2ROCK1GUSBDHODHBLM
SCHEMBL7148341 0.69 GUSB (0.55) ROCK2ROCK1GUSBDHODHBLM
SCHEMBL6154382 0.69 GUSB (0.40) ROCK2ROCK1GUSBDHODHBLM
SCHEMBL6153748 0.68 GUSB (0.54) ROCK2ROCK1GUSBBLMKMT2A
SCHEMBL6153683 0.68 GUSB (0.51) ROCK2ROCK1GUSBDHODHBLM
SCHEMBL6153810 0.68 KMO (0.55) ROCK2ROCK1GUSBDHODHBLM
SCHEMBL6153833 0.68 GUSB (0.48) GUSBBLMKMT2AKDM4EMEN1
SCHEMBL6154890 0.67 DHODH (0.44) ROCK2ROCK1GUSBDHODHBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1446110-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES Structural Bioinformatics Inc. (US) 2004-08-18 EP disclosed
WO-2003032916-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES STRUCTURAL BIOINFORMATICS INC. (US) 2003-04-24 WO disclosed