SCHEMBL6685197

SCHEMBL6685197

O=C(O)CCCCSC(=S)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.53
HDAC4 P56524 3/20 0.53
HDAC1 Q13547 3/20 0.53
HDAC7 Q8WUI4 3/20 0.53
HDAC2 Q92769 3/20 0.53
HDAC10 Q969S8 3/20 0.53
HDAC11 Q96DB2 3/20 0.53
HDAC8 Q9BY41 3/20 0.53
HDAC6 Q9UBN7 3/20 0.53
HDAC9 Q9UKV0 3/20 0.53
HDAC5 Q9UQL6 3/20 0.53
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.44
RXFP1 Q9HBX9 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
LMNA P02545 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NR4A2 P43354 1/20 0.44
PPARA Q07869 1/20 0.44
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15669215 0.95 ALDH1A1 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL18496979 0.87 CYP1A2 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL16972073 0.77 ALDH1A1 (0.46) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8308737 0.77 ALDH1A1 (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL10913857 0.77 NPSR1 (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL15669260 0.76 HDAC3 (0.35) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL15669258 0.76 HDAC3 (0.35) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL162936 0.76 ALDH1A1 (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4832150 0.74 ALDH1A1 (0.50) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4437686 0.73 ALDH1A1 (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11708446-B2 Polymers and uses thereof MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2023-07-25 US claimed
EP-3976878-A1 METHODS OF MAKING A DEFLECTION MEMBER The Procter & Gamble Company (US) 2022-04-06 EP claimed
WO-2020243748-A1 METHODS OF MAKING A DEFLECTION MEMBER THE PROCTER & GAMBLE COMPANY (US) 2020-12-03 WO claimed
WO-2024059936-A1 THREE-DIMENSIONAL SURFACE PATTERNING NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2024-03-28 WO disclosed
WO-2023244814-A1 POLYMER/CELLULOSE NANOCRYSTAL-BASED NANOCOMPOSITE AND METHOD OF MAKING SAME FOX DOUGLAS (US) 2023-12-21 WO disclosed
EP-4031173-A1 COMPOUNDS FOR THE INDUCTION OF ANTIGEN-SPECIFIC IMMUNE TOLERANCE Anokion SA (CH) 2022-07-27 EP disclosed
EP-3976878-A1 METHODS OF MAKING A DEFLECTION MEMBER The Procter & Gamble Company (US) 2022-04-06 EP disclosed
WO-2021083997-A1 NOVEL MICELLAR CATALYSTS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2021-05-06 WO disclosed
WO-2021053589-A1 COMPOUNDS FOR THE INDUCTION OF ANTIGEN-SPECIFIC IMMUNE TOLERANCE ANOKION SA (CH) 2021-03-25 WO disclosed
WO-2020243748-A1 METHODS OF MAKING A DEFLECTION MEMBER THE PROCTER & GAMBLE COMPANY (US) 2020-12-03 WO disclosed
EP-3710061-A1 POLYMER PRODRUGS AND SUBCUTANEOUS AND/OR INTRAMUSCULAR ADMINISTRATION THEREOF Centre National de la Recherche Scientifique (FR) 2020-09-23 EP disclosed
EP-3442594-A1 BLOCK COPOLYMER FOR OVERCOMING DRUG RESISTANCE OF TUMOURS TO CHEMOTHERAPY, ITS POLYMER-DRUG CONJUGATE, PHARMACEUTICAL COMPOSITION CONTAINING THEM, METHOD OF PREPARATION AND USE THEREOF Ustav Makromolekularni Chemie AV CR, v.v.i. (CZ) 2019-02-20 EP disclosed
WO-2018015222-A1 PROCESS BP EXPLORATION OPERATING COMPANY LIMITED (GB) 2018-01-25 WO disclosed
WO-2017218520-A1 SURFACE-COATED CONTINUOUS GLUCOSE MONITORS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2017-12-21 WO disclosed
WO-2017177991-A1 BLOCK COPOLYMER FOR OVERCOMING DRUG RESISTANCE OF TUMOURS TO CHEMOTHERAPY, ITS POLYMER-DRUG CONJUGATE, PHARMACEUTICAL COMPOSITION CONTAINING THEM, METHOD OF PREPARATION AND USE THEREOF USTAV MAKROMOLEKULARNI CHEMIE AV CR, V.V.I. (CZ) 2017-10-19 WO disclosed
WO-2016085535-A1 MODIFIED HETEROPHASIC POLYOLEFIN COMPOSITION MILLIKEN & COMPANY (US) 2016-06-02 WO disclosed
EP-2793581-A1 NANOPARTICLES COMPOSITIONS CONTAINING POLYMERS AND ANTHRANILIC ACID DIAMIDE INSECTICIDES FOR PROPAGULE COATING E. I. Du Pont de Nemours and Company (US) 2014-10-29 EP disclosed
WO-2014152850-A1 DENSELY FUNCTIONALIZED POLYMERS DERIVED FROM BAYLIS-HILLMAN ADDUCTS THE UNIVERSITY OF AKRON (US) 2014-09-25 WO disclosed
WO-2013096497-A1 NANOPARTICLES COMPOSITIONS CONTAINING POLYMERS AND ANTHRANILIC ACID DIAMIDE INSECTICIDES FOR PROPAGULE COATING E. I. DU PONT DE NEMOURS AND COMPANY (US) 2013-06-27 WO disclosed
WO-2004056880-A1 PROCESS FOR THE PREPARATION OF A MULTIBLOCK COPOLYMER STICHTING DUTCH POLYMER INSTITUTE (NL) 2004-07-08 WO disclosed