SCHEMBL6685864

SCHEMBL6685864

Cc1cc(CN[C@@H](C)C(N)=O)ccc1OCc1ccc(SC(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.46
SCN9A Q15858 2/20 0.46
MAOA P21397 1/20 0.46
CD274 Q9NZQ7 2/20 0.46
FFAR1 O14842 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43
PPARA Q07869 2/20 0.42
PTPRZ1 P23471 1/20 0.41
HRH3 Q9Y5N1 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6685862 1.00 MAOB (0.46) MAOBSCN9AMAOACD274FFAR1
SCHEMBL6685304 0.89 CD274 (0.42) CD274FFAR1FFAR4PPARAPTPRZ1
SCHEMBL6685310 0.89 CD274 (0.42) CD274FFAR1FFAR4PPARAPTPRZ1
SCHEMBL6693062 0.89 MAOB (0.45) MAOBSCN9AMAOACD274FFAR4
SCHEMBL6693067 0.89 MAOB (0.45) MAOBSCN9AMAOACD274FFAR4
SCHEMBL6685530 0.85 FFAR4 (0.48) CD274FFAR1FFAR4PPARA
SCHEMBL6685527 0.85 FFAR4 (0.48) CD274FFAR1FFAR4PPARA
SCHEMBL6688691 0.85 PDCD1 (0.44) MAOBSCN9AMAOACD274
SCHEMBL6685877 0.84 MAOB (0.61) MAOBSCN9AMAOAPTPRZ1HRH3
SCHEMBL6685873 0.84 MAOB (0.61) MAOBSCN9AMAOAPTPRZ1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed