SCHEMBL6693067

SCHEMBL6693067

COc1cc(CN[C@@H](C)C(N)=O)ccc1OCc1ccc(SC(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.45
MAOA P21397 2/20 0.45
SCN9A Q15858 2/20 0.45
FFAR4 Q5NUL3 1/20 0.44
NPC1 O15118 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
PDCD1 Q15116 2/20 0.42
CD274 Q9NZQ7 2/20 0.42
NTRK1 P04629 1/20 0.42
CSF1R P07333 1/20 0.42
NTRK2 Q16620 1/20 0.42
ALDH1A1 P00352 1/20 0.42
F2 P00734 1/20 0.42
F10 P00742 1/20 0.42
PRSS1 P07477 1/20 0.42
F7 P08709 1/20 0.42
MRGPRX1 Q96LB2 1/20 0.42
PTPRZ1 P23471 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6693062 1.00 MAOB (0.45) MAOBMAOASCN9AFFAR4NPC1
SCHEMBL6685506 0.89 PDCD1 (0.53) FFAR4NPC1PKMRAB9APDCD1
SCHEMBL6685503 0.89 PDCD1 (0.53) FFAR4NPC1PKMRAB9APDCD1
SCHEMBL6690103 0.89 ATM (0.47) FFAR4NPC1PKMRAB9APDCD1
SCHEMBL6690101 0.89 ATM (0.47) FFAR4NPC1PKMRAB9APDCD1
SCHEMBL6685289 0.89 FFAR4 (0.43) FFAR4NPC1PKMRAB9APDCD1
SCHEMBL6685286 0.89 FFAR4 (0.43) FFAR4NPC1PKMRAB9APDCD1
SCHEMBL6685862 0.89 MAOB (0.46) MAOBMAOASCN9AFFAR4CD274
SCHEMBL6685864 0.89 MAOB (0.46) MAOBMAOASCN9AFFAR4CD274
SCHEMBL6687571 0.87 MAOB (0.47) MAOBMAOASCN9ANPC1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed