SCHEMBL6686477

SCHEMBL6686477

CC(C)(C)CCn1c(=O)c(C2=NS(=O)(=O)c3cc(O)ccc3N2)c(O)c2cc(F)ccc21

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.63
NR1I2 O75469 1/20 0.63
MAPK1 P28482 1/20 0.49
HSD17B10 Q99714 1/20 0.49
PLK1 P53350 1/20 0.35
PTGDR2 Q9Y5Y4 6/20 0.34
PER2 O15055 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CRY1 Q16526 1/20 0.33
CRY2 Q49AN0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6685191 0.90 CYP2C9 (0.64) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6686456 0.89 HSD17B10 (0.61) CYP2C9NR1I2MAPK1HSD17B10L3MBTL1
SCHEMBL6732332 0.88 CYP2C9 (0.61) CYP2C9NR1I2MAPK1HSD17B10PTGDR2
SCHEMBL6690316 0.87 CYP2C9 (0.83) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6738466 0.86 CYP2C9 (0.63) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6692294 0.86 CYP2C9 (0.80) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6740621 0.83 CYP2C9 (0.57) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6738280 0.82 CYP2C9 (0.65) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6693468 0.81 CYP2C9 (0.81) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6732912 0.81 MAPK1 (0.57) CYP2C9NR1I2MAPK1HSD17B10PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004052312-A2 ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-06-24 WO disclosed