SCHEMBL6686492

SCHEMBL6686492

CCOC(=O)[C@@H](C)Oc1ccc2c(c1)S(=O)(=O)N=C(c1c(O)c3cc(F)ccc3n(CCC3CC3)c1=O)N2

nearest known ligand 0.85

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.85
NR1I2 O75469 1/20 0.68
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PLK1 P53350 2/20 0.35
HIF1A Q16665 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CRY1 Q16526 5/20 0.31
CRY2 Q49AN0 5/20 0.31
MKNK2 Q9HBH9 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
PER2 O15055 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6686493 1.00 CYP2C9 (0.85) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6688520 0.92 CYP2C9 (0.88) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6688517 0.92 CYP2C9 (0.88) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6738653 0.92 CYP2C9 (1.00) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6231450 0.92 CYP2C9 (1.00) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6684922 0.91 CYP2C9 (0.86) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6693133 0.91 CYP2C9 (0.86) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6689881 0.88 CYP2C9 (0.73) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6236224 0.88 CYP2C9 (0.80) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6680076 0.88 CYP2C9 (0.85) CYP2C9NR1I2MAPK1HSD17B10PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004052312-A2 ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-06-24 WO claimed
WO-2004052312-A2 ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-06-24 WO disclosed